3zrk A 2.37 BS02 ZRK A 1 V70 A83 K85 Y134 V135 L188 D200 V35 A48 K50 Y97 V98 L151 D163 D181 K183 N186 D200 S219 D144 K146 N149 D163 S182 2.7.11.1,2.7.11.26 0004672,0005524,0006468 ic50=0.13uM -logKd/Ki=6.89, IC50=0.13uM IC50=125.89nM P49841 21764580 1400 KVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSKKDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNYTEFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHARI 3zrk B 2.37 BS02 ZRK B 1 V70 A83 K85 Y134 V135 L188 D200 V35 A48 K50 Y99 V100 L153 D165 D181 K183 N186 D200 S219 D146 K148 N151 D165 S184 2.7.11.1,2.7.11.26 0004672,0005524,0006468 ic50=0.13uM IC50=125.89nM P49841 21764580 1400 KVTTVVATPGQGPDRPQEVSYTDTKVIGNGSFGVVYQAKLCDSGELVAIKKVLQDKRFKNRELQIMRKLDHCNIVRLRYFFYSSGEKKDEVYLNLVLDYVPETVYRVARHYSRAKQTLPVIYVKLYMYQLFRSLAYIHSFGICHRDIKPQNLLLDPDTAVLKLCDFGSAKQLVRGEPNVSYICSRYYRAPELIFGATDYTSSIDVWSAGCVLAELLLGQPIFPGDSGVDQLVEIIKVLGTPTREQIREMNPNYTEFKFPQIKAHPWTKVFRPRTPPEAIALCSRLLEYTPTARLTPLEACAHSFFDELRDPNVKLPNGRDTPALFNFTTQELSSNPPLATILIPPHARI