4ynk A 2.3 BS02 YW2 A 1 Y143 A227 V230 S233 R270 S271 S274 W282 Y291 H301 L309 H393 L410 Y21 A46 V49 S52 R89 S90 S93 W101 Y110 H120 L128 H212 L229 ? 0003677,0004879,0006355 -logKd/Ki=8.30, IC50=5nM P13053 26613420 500 KLSEEQQHIIAILLDAHHKTYDPTYADFRDFRPPVRMPLSMLPHLADLVSYSIQKVIGFAKMIPGFRDLTSDDQIVLLKSSAIEVIMLRSNQSFTMDDMSWDCGSQDYKYDVTDVSKAGHTLELIEPLIKFQVGLKKLNLHEEEHVLLMAICIVSPDRPGVQDAKLVEAIQDRLSNTLQTYIRCRHPPPGSHQLYAKMIQKLADLRSLNEEHSKQYRSLSFQPENSMKLTPLVLEVFGNE