4anb A 2.2 BS01 YQY A 1 K97 V127 I141 D208 F209 V211 L215 K40 V70 I84 D151 F152 V154 L158 D190 K192 S194 N195 D208 D217 T226 D133 K135 S137 N138 D151 D160 T169 2.7.12.2 0004672,0005524,0006468 -logKd/Ki=8.18, IC50=6.6nM IC50=6.6nM Q02750 24900486 501 MALGELKDDDFEKISELGAGNGGVVFKVSHKPSGLVMARKLIHLEIKPAIRNQIIRELQVLHECNSPYIVGFYGAFYSDGEISICMEHMDGGSLDQVLKKAGRIPEQILGKVSIAVIKGLTYLREKHKIMHRDVKPSNILVNSRGEIKLCDFGVSGQLIDEMANEFVGTRSYMSPERLQGTHYSVQSDIWSMGLSLVEMAVGRYPRPPMAIFELLDYIVNEPPPKLPSAVFSLEFQDFVNKCLIKNPAERADLKQLMVHAFIKRSDAEEVDFAGWLCSTIGL