5fto A 2.22 BS01 YMX A 1 L1122 G1123 F1127 V1130 A1148 L1196 M1199 A1200 G1202 D1203 N1254 L1256 G1269 L30 G31 F35 V38 A52 L100 M103 A104 G106 D107 N158 L160 G173 D1249 A1251 R1253 N1254 D1270 R1279 D153 A155 R157 N158 D174 R183 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 Ki=6.2nM -logKd/Ki=8.21, Ki=6.2nM IC50=55nM, Ki=6.2nM Q9UM73 27003761 2402 GPNYCFAGKTSSISDLKEVPRKNITLIRGLGHGAFGEVYEGQVSGMSPLQVAVKTLPEVCSEQDELDFLMEALIISKFNHQNIVRCIGVSLQSLPRFILLELMAGGDLKSFLRETRPRPSQPSSLAMLDLLHVARDIACGCQYLEENHFIHRDIAARNCLLTCPGPGRVAKIGDFGMARDIYRGCAMLPVKWMPPEAFMEGIFTSKTDTWSFGVLLWEIFSLGYMPYPSKSNQEVLEFVTSGGRMDPPKNCPGPVYRIMTQCWQHQPEDRPNFAIILERIEYCTQDPDVINTALPIEY 5kvt A 2.45 BS01 YMX A 1 L516 V524 A542 F589 M592 G595 D596 R599 N655 L657 G667 L16 V24 A38 F85 M88 G91 D92 R95 N151 L153 G163 D650 R654 N655 D668 D146 R150 N151 D164 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169,0016020 IC50=0.600nM P04629 801 CVHHIKRRDIVLKWELGEGAFGKVFLAECHNLDKMLVAVKALKEASESARQDFQREAELLTMLQHQHIVRFFGVCTEGRPLLMVFEYMRHGDLNRFLRSHGPDAKLLAGGEDVAPGPLGLGQLLAVASQVAAGMVYLAGLHFVHRDLATRNCLVGQGLVVKIGDFGMSRDIYSTDYYRVGGRTMLPIRWMPPESILYRKFTTESDVWSFGVVLWEIFTYGKQPWYQLSNTEAIDCITQGRELERPRACPPEVYAIMRGCWQREPQQRHSIKDVHARLQALAQAHHHH