2ym3 A 2.007 BS01 YM3 A 1 L15 G16 V23 A36 E85 Y86 C87 G90 E91 L137 L8 G9 V11 A24 E62 Y63 C64 G67 E68 L114 D130 K132 E134 N135 D148 T170 D107 K109 E111 N112 D125 T147 2.7.11.1 0000077,0004672,0004674,0005524,0006468 ic50=1.2uM -logKd/Ki=6.00, IC50=1.0uM IC50=1200nM O14757 22111927 1271 DWDLVQTLGEVQLAVNRVTEEAVAVKIVDNIKKEICINKMLNHENVVKFYGHRREIQYLFLEYCSGGELFDRIEPDIGMPEPDAQRFFHQLMAGVVYLHGIGITHRDIKPENLLLDERDNLKISDFGLATVFRYNNRERLLNKMCGTLPYVAPELLKRREFHAEPVDVWSCGIVLTAMLAGELPWDQPSDSCQEYSDWKEKKTYLNPWKKIDSAPLALLHKILVENPSARITIPDIKKDRWYNKPLK