5jv1 F 2.3 BS01 YL6 F 1 K57 N59 R60 S205 F206 F239 Q242 D243 K45 N47 R48 S191 F192 F225 Q228 D229 2.5.1.1,2.5.1.10 0004659,0008299,0016765 ic50=0.86uM -logKd/Ki=6.07, IC50=0.86uM P14324 28208018 403 VYAQEKQDFVQHFSQIVRVLTEHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 5jv1 F 2.3 BS02 YL6 F 2 E319 Y322 A345 R346 Y349 K350 E305 Y308 A331 R332 Y335 K336 2.5.1.1,2.5.1.10 0004659,0008299,0016765 ic50=0.86uM -logKd/Ki=6.07, IC50=0.86uM P14324 28208018 404 VYAQEKQDFVQHFSQIVRVLTEHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK 6n83 F 2.0 BS01 YL6 F 1 N59 R60 S205 F206 F239 Q242 L344 N50 R51 S196 F197 F230 Q233 L335 K57 F98 D103 D107 R112 D174 K200 F239 D243 D244 K48 F89 D94 D98 R103 D165 K191 F230 D234 D235 2.5.1.1,2.5.1.10 0004659,0008299,0016765 ic50=0.54uM -logKd/Ki=6.27, IC50=0.54uM P14324 31577901 401 SDVYAQEKQDFVQHFSQIVRVLTEGHPEIGDAIARLKEVLEYNAIGGKYNRGLTVVVAFRELVEPRKQDADSLQRAWTVGWCVELLQAFFLVADDIMDSSLTRRGQICWYQKPGVGLDAINDANLLEACIYRLLKLYCREQPYYLNLIELFLQSSYQTEIGQTLDLLTAPQGNVDLVRFTEKRYKSIVKYKTAFYSFYLPIAAAMYMAGIDGEKEHANAKKILLEMGEFFQIQDDYLDLFGDPSVTGKIGTDIQDNKCSWLVVQCLQRATPEQYQILKENYGQKEAEKVARVKALYEELDLPAVFLQYEEDSYSHIMALIEQYAAPLPPAVFLGLARKIYK