2y5k A 2.1 BS01 YCU A 1 M18 G21 R22 G26 G28 L30 T31 M177 D178 M10 G13 R14 G18 G20 L22 T23 M161 D162 D74 E97 E98 D118 L120 D121 E280 D58 E81 E82 D102 L104 D105 E264 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0005986,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 ic50=0.22uM -logKd/Ki=6.66, IC50=0.22uM IC50=220nM P09467 21550236 1336 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGVKKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 2y5k A 2.1 BS02 YCU C 1 T27 G28 T19 G20 D74 E97 E98 D118 L120 D121 E280 D58 E81 E82 D102 L104 D105 E264 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0005986,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 ic50=0.22uM -logKd/Ki=6.66, IC50=0.22uM IC50=220nM P09467 21550236 1336 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGVKKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 2y5k B 2.1 BS01 YCU B 1 V17 M18 G21 R22 G26 G28 L30 T31 V9 M10 G13 R14 G18 G20 L22 T23 D74 E97 E98 D118 L120 D121 E280 D56 E79 E80 D100 L102 D103 E262 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0005986,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 ic50=0.22uM IC50=220nM P09467 21550236 1336 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 2y5k C 2.1 BS01 YCU A 1 T27 T31 T19 T23 D74 E97 E98 D118 L120 D121 E280 D57 E80 E81 D101 L103 D104 E263 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0005986,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 ic50=0.22uM -logKd/Ki=6.66, IC50=0.22uM IC50=220nM P09467 21550236 1336 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGKKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 2y5k C 2.1 BS02 YCU C 1 M18 G21 R22 G26 G28 L30 T31 M177 D178 M10 G13 R14 G18 G20 L22 T23 M160 D161 D74 E97 E98 D118 L120 D121 E280 D57 E80 E81 D101 L103 D104 E263 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0005986,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 ic50=0.22uM -logKd/Ki=6.66, IC50=0.22uM IC50=220nM P09467 21550236 1336 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGKKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 2y5k D 2.1 BS01 YCU B 1 T27 G28 T19 G20 D74 E97 E98 D118 L120 D121 E280 D56 E79 E80 D100 L102 D103 E262 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0005986,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 ic50=0.22uM IC50=220nM P09467 21550236 1336 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS 2y5k D 2.1 BS02 YCU D 1 V17 M18 G21 R22 G26 G28 L30 T31 V9 M10 G13 R14 G18 G20 L22 T23 D74 E97 E98 D118 L120 D121 E280 D56 E79 E80 D100 L102 D103 E262 3.1.3.11 0000122,0005515,0005615,0005634,0005737,0005829,0005975,0005986,0006000,0006002,0006094,0006111,0016208,0016311,0016787,0016791,0030308,0030388,0031667,0032869,0042132,0042578,0042802,0045820,0046580,0046872,0048029,0061629,0070062,0071286,0071320,0071466,0071475,0071477,0097403,1904628 ic50=0.22uM IC50=220nM P09467 21550236 1336 DVNTLTRFVMEEGRKARGTGELTQLLNSLCTAVKAISSAVRKAGIAHLYGIAGKLDVLSNDLVMNMLKSSFATCVLVSEEDKHAIIVEPEKRGKYVVCFDPLDGSSNIDCLVSVGTIFGIYRKKSTDEPSEKDALQPGRNLVAAGYALYGSATMLVLAMDCGVNCFMLDPAIGEFILVDKDVKIKKKGKIYSLNEGYAKDFDPAVTEYIQRKKFPPDNSAPYGARYVGSMVADVHRTLVYGGIFLYPANKKSPNGKLRLLYECNPMAYVMEKAGGMATTGKEAVLDVIPTDIHQRAPVILGSPDDVLEFLKVYEKHS