3pkc A 1.47 BS03 Y08 A 1 E35 Y97 H114 D131 D142 T203 H205 F211 H212 E238 E269 E32 Y94 H111 D128 D139 T200 H202 F208 H209 E235 E266 H114 D131 D142 G204 H205 G208 H212 L215 E238 N242 E269 H111 D128 D139 G201 H202 G205 H209 L212 E235 N239 E266 3.4.11.18 0004177,0004239,0005506,0005829,0006508,0008235,0016485,0046872,0046914,0050897,0070006 ic50=0.96uM -logKd/Ki=6.02, IC50=960nM P9WK19 21465667 288 RTALSPGVLSPTRPVPNWIARPEYVGKPAAQEGSEPWVQTPEVIEKMRVAGRIAAGALAEAGKAVAPGVTTDELDRIAHEYLVDNGAYPSTLGYKGFPKSCCTSLNEVICHGIPDSTVITDGDIVNIDVTAYIGGVHGDTNATFPAGDVADEHRLLVDRTREATMRAINTVKPGRALSVIGRVIESYANRFGYNVVRDFTGHGIGTTFHNGLVVLHYDQPAVETIMQPGMTFTIEPMINLGALDYEIWDDGWTVVTKDRKWTAQFEHTLLVTDTGVEILTC 4flj A 1.74 BS03 Y08 A 1 Y195 H212 D229 D240 C301 H303 F309 H310 E336 E367 Y106 H123 D140 D151 C212 H214 F220 H221 E247 E278 D229 D240 H303 H310 E336 E367 D140 D151 H214 H221 E247 E278 3.4.11.18 0006508,0070006 ic50=7.45uM -logKd/Ki=5.13, IC50=7.45uM P53582 22913487 503 YRYTGKLRPHYPLMPTRPVPSYIQRPDYADHPLGMSESEQALKGTSQIKLLSSEDIEGMRLVCRLAREVLDVAAGMIKPGVTTEEIDHAVHLACIARNCYPSPLNYYNFPKSCCTSVNEVICHGIPDRRPLQEGDIVNVDITLYRNGYHGDLNETFFVGEVDDGARKLVQTTYECLMQAIDAVKPGVRYRELGNIIQKHAQANGFSVVRSYCGHGIHKLFHTAPNVPHYAKNKAVGVMKSGHVFTIEPMICEGGWQDETWPDGWTAVTRDGKRSAQFEHTLLVTDTGCEILTRRLDSARPHFMS