4eqc A 2.01 BS01 XR1 A 1 A297 R299 E315 V342 M344 Y346 L347 G350 L396 T541 A53 R55 E71 V98 M100 Y102 L103 G106 L152 T297 D389 K391 D393 N394 D407 P416 T427 D145 K147 D149 N150 D163 P172 T183 2.7.11.1 0004672,0005524,0006468 ic50=8nM -logKd/Ki=8.10, IC50=8nM IC50=2.8nM Q13153 23960073 601 DPFTSDEEILEKLRSIVSVGDPKKKYTRFEKIGQGASGTVYTAMDVATGQEVAIRQMNLQQQPKKELIINEILVMRENKNPNIVNYLDSYLVGDELWVVMEYLAGGSLTDVVTETCMDEGQIAAVCRECLQALEFLHSNQVIHRDIKSDNILLGMDGSVKLTDFGFCAQITPEQSKRSTMVGTPYWMAPEVVTRKAYGPKVDIWSLGIMAIEMIEGEPPYLNENPLRALYLIATNGTPELQNPEKLSAIFRDFLNRCLEMDVEKRGSAKELLQHQFLKIAKPLSSLTPLIAAAKEAT