3q92 A 2.8 BS01 XNB A 1 A224 A226 E227 G229 P246 V250 G257 F260 C282 A222 A224 E225 G227 P244 V248 G255 F258 C280 G255 A256 G257 D258 G253 A254 G255 D256 2.7.1.3 0004454,0005515,0005524,0005737,0005829,0006000,0006796,0009744,0009749,0009750,0010043,0016301,0016310,0032868,0042802,0042803,0046835,0070061,0070062,0070873 -logKd/Ki=7.92, IC50=12nM IC50=<500nM P50053 24900346 301 GSQILCVGLVVLDVISLVDKYPKEDSEIRCLSQRWQRGGNASNSCTVLSLLGAPCAFMGSMAPGHVADFLVADFRRRGVDVSQVAWQSKGDTPSSCCIINNSNGNRTIVLHDTSLPDVSATDFEKVDLTQFKWIHIEGRNASEQVKMLQRIDAHNTRQPPEQKIRVSVEVEKPREELFQLFGYGDVVFVSKDVAKHLGFQSAEEALRGLYGRVRKGAVLVCAWAEEGADALGPDGKLLHSDAFPPPRVVDTLGAGDTFNASVIFSLSQGRSVQEALRFGCQVAGKKCGLQGFDGIV 3q92 B 2.8 BS01 XNB B 1 A226 G229 F245 P246 V250 G257 F260 C289 A229 G232 F248 P249 V253 G260 F263 C292 G255 A256 G257 D258 G258 A259 G260 D261 2.7.1.3 0004454,0005515,0005524,0005737,0005829,0006000,0006796,0009744,0009749,0009750,0010043,0016301,0016310,0032868,0042802,0042803,0046835,0070061,0070062,0070873 -logKd/Ki=7.92, IC50=12nM IC50=<500nM P50053 24900346 301 GLVPRGSQILCVGLVVLDVISLVDKYPKEDSEIRCLSQRWQRGGNASNSCTVLSLLGAPCAFMGSMAPGHVADFLVADFRRRGVDVSQVAWQSKGDTPSSCCIINNSNGNRTIVLHDTSLPDVSATDFEKVDLTQFKWIHIEGRNASEQVKMLQRIDAHNTRQPPEQKIRVSVEVEKPREELFQLFGYGDVVFVSKDVAKHLGFQSAEEALRGLYGRVRKGAVLVCAWAEEGADALGPDGKLLHSDAFPPPRVVDTLGAGDTFNASVIFSLSQGRSVQEALRFGCQVAGKKCGLQGFDGIV