2xk9 A 2.35 BS01 XK9 A 1 L226 V234 K249 I251 E273 L301 M304 E305 G307 L354 T367 D368 L16 V23 K38 I40 E47 L75 M78 E79 G81 L128 T141 D142 D347 K349 N352 D368 T387 D121 K123 N126 D142 T161 2.7.11.1 0004672,0005524,0006468 ic50=0.03nM -logKd/Ki=10.15, IC50=0.07nM O96017 21963792 1511 VYPKALRDEYIMSKTLGSGAGEVKLAFERKTCKKVAIKIISKNVETEIEILKKLNHPCIIKIKNFFDAEDYYIVLELMEGGELFDKVVGNKRLKEATCKLYFYQMLLAVQYLHENGIIHRDLKPENVLLSSQEEDCLIKITDFGHSKILGETSLMRTLCGTPTYLAPEVLVSVGTAGYNRAVDCWSLGVILFICLSGYPPFSEHRTQVSLKDQITSGKYNFIPEVWAEVSEKALDLVKKLLVVDPKARFTTEEALRHPWLQDEDMKRKFQDLLSEENESTALPQ