1j3i A 2.33 BS01 WRA A 1 I14 C15 D54 M55 F58 P113 F116 I164 I14 C15 D54 M55 F58 P103 F106 I154 L46 D54 L46 D54 1.5.1.3,2.1.1.45 0004146,0046654,0050661 Ki=0.011nM IC50=0.570000nM, Ki=0.5nM P13922 12704428 609 MMEQVCDVFDIYAICACCKVESKNEGKKNEVFNNYTFRGLGNKGVLPWKCNSLDMKYFCAVTTYVNESKYEKLKYKRCKYLNKETKKLQNVVVMGRTSWESIPKKFKPLSNRINVILSRTLKKEDFDEDVYIINKVEDLIVLLGKLNYYKCFIIGGSVVYQEFLEKKLIKKIYFTRINSTYECDVFFPEINENEYQIISVSDVYTSNNTTLDFIIYKKTNNKM 1j3i B 2.33 BS01 WRA B 1 I14 C15 L46 D54 M55 F58 P113 I164 I13 C14 L45 D53 M54 F57 P108 I159 L46 D54 L45 D53 1.5.1.3,2.1.1.45 0004146,0046654,0050661 Ki=0.011nM IC50=0.570000nM, Ki=0.5nM P13922 12704428 709 MEQVCDVFDIYAICACCKVESKNEGKKNEVFNNYTFRGLGNKGVLPWKCNSLDMKYFCAVTTYVNESKYEKLKYKRCKYLNKETVDMPNSKKLQNVVVMGRTSWESIPKKFKPLSNRINVILSRTLKKEDFDEDVYIINKVEDLIVLLGKLNYYKCFIIGGSVVYQEFLEKKLIKKIYFTRINSTYECDVFFPEINENEYQIISVSDVYTSNNTTLDFIIYKKTNN 1j3k A 2.1 BS01 WRA A 1 I14 C15 D54 M55 F58 N108 P113 I14 C15 D54 M55 F58 N98 P103 L46 D54 L46 D54 1.5.1.3,2.1.1.45 0004146,0046654,0050661 Ki=0.037nM IC50=0.570000nM, Ki=0.5nM P13922 12704428 609 MMEQVCDVFDIYAICACCKVESKNEGKKNEVFNNYTFRGLGNKGVLPWKCISLDMKYFRAVTTYVNESKYEKLKYKRCKYLNKETKKLQNVVVMGRTNWESIPKKFKPLSNRINVILSRTLKKEDFDEDVYIINKVEDLIVLLGKLNYYKCFILGGSVVYQEFLEKKLIKKIYFTRINSTYECDVFFPEINENEYQIISVSDVYTSNNTTLDFIIYKKTNN 1j3k B 2.1 BS01 WRA B 1 I14 C15 D54 M55 F58 N108 P113 I14 C15 D54 M55 F58 N97 P102 L46 D54 L46 D54 1.5.1.3,2.1.1.45 0004146,0046654,0050661 Ki=0.037nM IC50=0.570000nM, Ki=0.5nM P13922 12704428 709 MMEQVCDVFDIYAICACCKVESKNEGKKNEVFNNYTFRGLGNKGVLPWKCISLDMKYFRAVTTYVNESKYEKLKYKRCKYLPNSKKLQNVVVMGRTNWESIPKKFKPLSNRINVILSRTLKKEDFDEDVYIINKVEDLIVLLGKLNYYKCFILGGSVVYQEFLEKKLIKKIYFTRINSTYECDVFFPEINENEYQIISVSDVYTSNNTTLDFIIYKKTNNK 3rg9 A 2.0 BS02 WRA A 1 V32 V33 I47 D54 M55 F58 T86 L90 P91 I160 V10 V11 I25 D32 M33 F36 T64 L68 P69 I138 I47 D54 I25 D32 1.5.1.3,2.1.1.45 0004146,0046654,0050661 Ki=1.1nM Q27783 21650210 602 RPPLRPFSVVVASDEKGGIGDGGTIPWEIPEDMQYFRRVTTNLRGKNVKPSPSKRNAVVMGRKTWDSLPPKFRPLSNRLNVVLSRSATKEQLLAGIPDPIKRAEAANDVVAVNGGLEDALRMLVSKEHTSSIETVFCIGGGTIYKQALCAPCVNVLQAIHRTVVRPASNSCSVFFDIPAAGTKTPEGLELVRESITDERVSTGAGGKKYQFEKLVPRN 3rg9 B 2.0 BS02 WRA B 1 V32 V33 I47 D54 M55 F58 T86 L90 P91 F94 I160 V10 V11 I25 D32 M33 F36 T64 L68 P69 F72 I138 I47 D54 I25 D32 1.5.1.3,2.1.1.45 0004146,0046654,0050661 Ki=1.1nM Q27783 21650210 702 RPPLRPFSVVVASDEKGGIGDGGTIPWEIPEDMQYFRRVTTNLRGKNVKPSPSKRNAVVMGRKTWDSLPPKFRPLSNRLNVVLSRSATKEQLLAGIPDPIKRAEAANDVVAVNGGLEDALRMLVSKEHTSSIETVFCIGGGTIYKQALCAPCVNVLQAIHRTVVRPASNSCSVFFDIPAAGTKTPEGLELVRESITDERVSTGAGGKKYQFEKLVPRN