4yti A 2.52 BS01 VJK A 1 G856 V863 A880 E930 Y931 L932 R980 N981 L983 G993 D994 G15 V22 A39 E86 Y87 L88 R136 N137 L139 G149 D150 D976 A978 R980 N981 D994 S1016 D132 A134 R136 N137 D150 S172 2.7.10.2 0004672,0004713,0005524,0006468 -logKd/Ki=7.89, Ki=13nM IC50=>10000nM, Ki=13nM O60674 26230873 4000 TQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSRNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDNM