2wd7 A 1.9 BS02 VGD A 1 S95 F97 Y174 S94 F96 Y155 R14 D161 Y174 K178 R13 D142 Y155 K159 1.5.1.33 0000166,0016491,0047040 Ki=10.6uM -logKd/Ki=4.97, Ki=10.6uM Ki=10600nM O76290 19527033 1269 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVGKTVETQVAELIGTNAIAPFLLTMSFAQRQSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 2wd7 B 1.9 BS02 VGD B 1 S95 F97 Y174 S94 F96 Y154 R14 D161 Y174 K178 R13 D141 Y154 K158 1.5.1.33 0000166,0016491,0047040 Ki=10.6uM Ki=10600nM O76290 19527033 1269 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVGKTVETQVAELIGTNAIAPFLLTMSFAQRQNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 2wd7 C 1.9 BS02 VGD C 1 S95 F97 Y174 S94 F96 Y155 R14 D161 Y174 K178 R13 D142 Y155 K159 1.5.1.33 0000166,0016491,0047040 Ki=10.6uM Ki=10600nM O76290 19527033 1269 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVGKTVETQVAELIGTNAIAPFLLTMSFAQRQSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 2wd7 D 1.9 BS02 VGD D 1 S95 F97 Y174 S94 F96 Y155 R14 D161 Y174 K178 R13 D142 Y155 K159 1.5.1.33 0000166,0016491,0047040 Ki=10.6uM Ki=10600nM O76290 19527033 1269 EAPAAVVTGAAKRIGRAIAVKLHQTGYRVVIHYHNSAEAAVSLADELNKERSNTAVVCQADLTNSNVLPASCEEIINSCFRAFGRCDVLVNNASAFYPTPLVGKTVETQVAELIGTNAIAPFLLTMSFAQRQSNLSIVNLCDAMVDQPCMAFSLYNMGKHALVGLTQSAALELAPYGIRVNGVAPGVSLLPVAMGEEEKDKWRRKVPLGRREASAEQIADAVIFLVSGSAQYITGSIIKVDGGLSLVHA 3kr1 A 2.3 BS02 VGD A 1 Y35 N39 R44 V53 F182 M258 Y12 N16 R21 V30 F159 M235 2.1.1.28 0004603,0005515,0005829,0008168,0032259,0042418,0042423 Kd=1.8uM -logKd/Ki=5.74, Kd=1.8uM P11086 20642456 290 ASAYQRFEPRAYLRNNYAPPRGDLCNPNGVGPWKLRCLAQTFATGEVSGRTLIDIGSGPTVYQLLSACSHFEDITMTDFLEVNRQELGRWLQEEPGAFNWSMYSQHACLIEGKGECWQDKERQLRARVKRVLPIDVHQPQPLGAGSPAPLPADALVSAFCLEAVSPDLASFQRALDHITTLLRPGGHLLLIGALEESWYLAGEARLTVVPVSEEEVREALVRSGYKVRDLRTYIMPAHLQTGVDDVKGVFFAWAQKV 3kr1 B 2.3 BS02 VGD B 1 N39 R44 V53 F182 Y222 M258 N26 R31 V40 F169 Y209 M245 2.1.1.28 0004603,0005515,0005829,0008168,0032259,0042418,0042423 Kd=1.8uM P11086 20642456 290 PDSAPGQAAVASAYQRFEPRAYLRNNYAPPRGDLCNPNGVGPWKLRCLAQTFATGEVSGRTLIDIGSGPTVYQLLSACSHFEDITMTDFLEVNRQELGRWLQEEPGAFNWSMYSQHACLIEGKGECWQDKERQLRARVKRVLPIDVHQPQPLGAGSPAPLPADALVSAFCLEAVSPDLASFQRALDHITTLLRPGGHLLLIGALEESWYLAGEARLTVVPVSEEEVREALVRSGYKVRDLRTYIMPAHLQTGVDDVKGVFFAWAQKVG