3h06 B 2.8 BS01 VBP B 1 Y61 P89 L90 T91 R96 T143 L192 E193 Y220 Y57 P85 L86 T87 R92 T139 L188 E189 Y216 ? 0015276,0016020 IC50=290000nM P19491 19284741 807 TVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 3h06 E 2.8 BS01 VBP E 1 Y61 P89 L90 T91 R96 L138 T143 T174 E193 M196 Y220 Y57 P85 L86 T87 R92 L134 T139 T170 E189 M192 Y216 ? 0015276,0016020 IC50=290000nM P19491 19284741 808 TVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 3h06 G 2.8 BS01 VBP G 1 Y61 P89 T91 R96 L138 T143 E193 Y220 Y57 P85 T87 R92 L134 T139 E189 Y216 ? 0015276,0016020 -logKd/Ki=3.53, IC50=292uM IC50=290000nM P19491 19284741 803 TVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 3h06 H 2.8 BS01 VBP H 1 E13 Y61 P89 T91 R96 L138 T143 T174 E193 M196 E9 Y57 P85 T87 R92 L134 T139 T170 E189 M192 ? 0015276,0016020 IC50=290000nM P19491 19284741 806 TVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 3h06 J 2.8 BS01 VBP J 1 Y61 P89 L90 T91 R96 L138 T143 L192 E193 Y57 P85 L86 T87 R92 L134 T139 L188 E189 ? 0015276,0016020 IC50=290000nM P19491 19284741 804 TVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 3h06 L 2.8 BS01 VBP L 1 Y16 Y61 P89 L90 T91 R96 L138 T143 T174 L192 E193 M196 Y220 Y12 Y57 P85 L86 T87 R92 L134 T139 T170 L188 E189 M192 Y216 ? 0015276,0016020 IC50=290000nM P19491 19284741 801 TVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 3h06 N 2.8 BS01 VBP N 1 E13 Y61 P89 T91 R96 L138 T143 L192 E193 M196 E9 Y57 P85 T87 R92 L134 T139 L188 E189 M192 ? 0015276,0016020 IC50=290000nM P19491 19284741 802 TVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 3h06 P 2.8 BS01 VBP P 1 Y61 P89 L90 T91 R96 L138 T143 T174 L192 E193 M196 Y57 P85 L86 T87 R92 L134 T139 T170 L188 E189 M192 ? 0015276,0016020 IC50=290000nM P19491 19284741 805 TVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC