1o0m A 1.5 BS01 U2P A 1 Q11 H12 K41 V43 N44 T45 H119 F120 Q11 H12 K41 V43 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=7.1uM -logKd/Ki=5.15, Ki=7.1uM Ki=11600nM P61823 14573867 1101 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 1o0m B 1.5 BS01 U2P B 1 Q11 H12 N44 T45 H119 F120 Q11 H12 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005515,0005576,0016829,0050830 Ki=7.1uM Ki=11600nM P61823 14573867 1201 KETAAAKFERQHMDSSTSAASSSNYCNQMMKSRNLTKDRCKPVNTFVHESLADVQAVCSQKNVACKNGQTNCYQSYSTMSITDCRETGSSKYPNCAYKTTQANKHIIVACEGNPYVPVHFDASV 1uca A 1.48 BS01 U2P A 1 Q9 N71 V72 L73 F80 H83 K87 Q9 N71 V72 L73 F80 H83 K87 H34 W37 S44 E84 K87 H88 H34 W37 S44 E84 K87 H88 4.6.1.19 0003723,0004519,0004521,0005576,0006401,0016829,0033897 P23540 10964705 400 FDSFWFVQQWPPAVCSFQKSGSCPGSGLRTFTIHGLWPQQSGTSLTNCPGSPFDITKISHLQSQLNTLWPNVLRANNQQFWSHEWTKHGTCSESTFNQAAYFKLAVDMRNNYDIIGALRPHAAGPNGRTKSRQAIKGFLKAKFGKFPGLRCRTDPQTKVSYLVQVVACFAQDGSTLIDCTRDTCGANFIF 1vd3 A 1.8 BS01 U2P A 1 H39 W42 W50 H92 E93 K96 H97 H39 W42 W50 H92 E93 K96 H97 H39 W42 W50 E93 K96 H97 H39 W42 W50 E93 K96 H97 3.1.27.1 0003723,0033897 Q9SSV1 214 AQDFDFFYFVQQWPASYCDTRRSCCYPTTGKPDEDFSIHGLWPNYENGKWPQNCDRESSLDESEISDLISTMEKNWPSLACPSSDGVRFWSHEWLKHGTCSALGERAYFQAALDFRKKSNLLENLKNAEITPRNGEHYTLESIKKAIEEGVGHSPYIECNVDTQGNHQIYQVYLCVDKTATDFIDCPIFPHGRGCGSKIEFPPF 1z4j A 1.8 BS03 U2P A 1 N41 D43 F49 W76 V77 T130 S131 P132 I133 K165 N8 D10 F16 W43 V44 T97 S98 P99 I100 K132 N41 D43 D176 N8 D10 D143 3.1.3.- 0008253,0009264 Q9NPB1 16004879 3001 RALRVLVNMDGVLADFEGGFLRKFRARFPDQPFIALEDRRGFWVSEQYGRLRPGLSEKAISIWESKNFFFELEPLPGAVEAVKEMASLQNTDVFICTSPIKMFKYCPYEKYAWVEKYFGPDFLEQIVLTRDKTVVSADLLIDDRPDITGAEPTPSWEHVLFTACHNQHLQLQPPRRRLHSWADDWKAILDSKRP 3djo A 1.6 BS01 U2P A 1 V43 N44 T45 K66 R85 F120 D121 V43 N44 T45 K66 R85 F120 D121 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005576,0016829,0042802,0050830,0051607 Ki=40.8uM -logKd/Ki=4.39, Ki=40.8uM Ki=40800nM P00669 19643512 125 KESAAAKFERQHMDSGNSPSSSSNYCNLMMCCRKMTQGKCKPVNTFVHESLADVKAVCSQKKVTCKNGQTNCYQSKSTMRITDCRETGSSKYPNCAYKTTQVEKHIIVACGGKPSVPVHFDASV 3djo A 1.6 BS02 U2P B 1 Q11 H12 Q11 H12 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005576,0016829,0042802,0050830,0051607 Ki=40.8uM -logKd/Ki=4.39, Ki=40.8uM Ki=40800nM P00669 19643512 201 KESAAAKFERQHMDSGNSPSSSSNYCNLMMCCRKMTQGKCKPVNTFVHESLADVKAVCSQKKVTCKNGQTNCYQSKSTMRITDCRETGSSKYPNCAYKTTQVEKHIIVACGGKPSVPVHFDASV 3djo B 1.6 BS01 U2P B 1 K41 V43 N44 T45 H119 F120 K41 V43 N44 T45 H119 F120 H12 K41 H119 F120 D121 H12 K41 H119 F120 D121 4.6.1.18 0003676,0004519,0004522,0004540,0005576,0016829,0042802,0050830,0051607 Ki=40.8uM -logKd/Ki=4.39, Ki=40.8uM Ki=40800nM P00669 19643512 201 KESAAAKFERQHMDSGNSPSSSSNYCNLMMCCRKMTQGKCKPVNTFVHESLADVKAVCSQKKVTCKNGQTNCYQSKSTMRITDCRETGSSKYPNCAYKTTQVEKHIIVACGGKPSVPVHFDASV 4dvn A 2.38 BS01 U2P A 1 H32 W35 H76 E77 K80 H81 H30 W33 H74 E75 K78 H79 2.7.7.48,3.4.21.113,3.4.22.-,3.6.1.15,3.6.4.13,4.6.1.19 0003723,0033897 Q96662 22579253 1118 ENITQWNLQDNGTEGIQRAMFQRGVNRSLHGIWPEKICTGVPSHLATDTELKAIHGMMDASEKTNYTCCRLQRHEWNKHGWCNWYNIEPWILLMNKTQANLTEGQPLRECAVTCRYDRDSDLNVVTQARDSPTPLTGCKKGKNFSFAGILVQGPCNFEIAV 4dvn A 2.38 BS02 U2P A 2 N9 H32 A62 Q129 N7 H30 A60 Q127 2.7.7.48,3.4.21.113,3.4.22.-,3.6.1.15,3.6.4.13,4.6.1.19 0003723,0033897 Q96662 22579253 1119 ENITQWNLQDNGTEGIQRAMFQRGVNRSLHGIWPEKICTGVPSHLATDTELKAIHGMMDASEKTNYTCCRLQRHEWNKHGWCNWYNIEPWILLMNKTQANLTEGQPLRECAVTCRYDRDSDLNVVTQARDSPTPLTGCKKGKNFSFAGILVQGPCNFEIAV 4dvn B 2.38 BS02 U2P B 1 N9 I18 Q19 H32 A62 N7 I16 Q17 H30 A60 2.7.7.48,3.4.21.113,3.4.22.-,3.6.1.15,3.6.4.13,4.6.1.19 0003723,0033897 Q96662 22579253 1113 ENITQWNLQDNGTEGIQRAMFQRGVNRSLHGIWPEKICTGVPSHLATDTELKAIHGMMDASEKTNYTCCRLQRHEWNKHGWCNWYNIEPWILLMNKTQANLTEGQPLRECAVTCRYDRDSDLNVVTQARDSPTPLTGCKKGKNFSFAGILVQGPCNFEIAV