2gg5 A 2.12 BS03 U19 A 1 Y62 Y65 D97 H171 F177 H178 E204 W221 Y61 Y64 D96 H170 F176 H177 E203 W220 H79 D97 D108 H171 R175 H178 Q182 E204 N208 Q233 E235 H78 D96 D107 H170 R174 H177 Q181 E203 N207 Q232 E234 3.4.11.18 0004177,0004239,0005829,0006508,0008198,0008235,0046872,0046914,0070006 ic50=0.25uM -logKd/Ki=6.60, IC50=0.25uM IC50=250nM P0AE18 17120228 501 AISIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGRGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISHDE