2gg7 A 1.12 BS03 U14 A 1 C59 Y62 H63 Y65 H79 D97 D108 H171 F177 H178 E204 W221 C58 Y61 H62 Y64 H78 D96 D107 H170 F176 H177 E203 W220 H79 D97 D108 H171 R175 H178 Q182 E204 N208 Q233 E235 H78 D96 D107 H170 R174 H177 Q181 E203 N207 Q232 E234 3.4.11.18 0004177,0004239,0005829,0006508,0008198,0008235,0046872,0046914,0070006 ic50=1.75uM -logKd/Ki=5.76, IC50=1.75uM IC50=1750nM P0AE18 17120228 701 AISIKTPEDIEKMRVAGRLAAEVLEMIEPYVKPGVSTGELDRICNDYIVNEQHAVSACLGYHGYPKSVCISINEVVCHGIPDDAKLLKDGDIVNIDVTVIKDGFHGDTSKMFIVGKPTIMGERLCRITQESLYLALRMVKPGINLREIGAAIQKFVEAEGFSVVREYCGHGIGRGFHEEPQVLHYDSRETNVVLKPGMTFTIEPMVNAGKKEIRTMKDGWTVKTKDRSLSAQYEHTIVVTDNGCEILTLRKDDTIPAIISHDE