3tza A 1.9 BS01 TZG A 1 Y58 P86 L87 T88 R93 L135 T140 E190 M193 Y60 P88 L89 T90 R95 L137 T142 E192 M195 ? 0015276,0016020 Ki=3.15uM -logKd/Ki=5.50, Ki=3.15uM P19491 21923187 261 ANKTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGECG 3tza B 1.9 BS01 TZG B 1 Y58 L87 T88 R93 L135 T140 E190 M193 Y217 Y58 L87 T88 R93 L135 T140 E190 M193 Y217 ? 0015276,0016020 Ki=3.15uM P19491 21923187 261 KTVVVTTILESPYVMMKKNHEMLEGNERYEGYCVDLAAEIAKHCGFKYKLTIVGDGKYGARDADTKIWNGMVGELVYGKADIAIAPLTITLVREEVIDFSKPFMSLGISIMIKKGTPIESAEDLSKQTEIAYGTLDSGSTKEFFRRSKIAVFDKMWTYMRSAEPSVFVRTTAEGVARVRKSKGKYAYLLESTMNEYIEQRKPCDTMKVGGNLDSKGYGIATPKGSSLGNAVNLAVLKLNEQGLLDKLKNKWWYDKGEC 4dld A 2.0 BS01 TZG A 1 Y16 Y61 P88 L89 T90 R95 S141 T142 S173 E190 S193 Y216 Y14 Y59 P86 L87 T88 R93 S139 T140 S171 E188 S191 Y214 ? 0015276,0016020 Ki=1.5uM -logKd/Ki=5.82, Ki=1.5uM Ki=3000nM P22756 22407805 301 NRTLIVTTILEEPYVMYRKSDKPLYGNDRFEGYCLDLLKELSNILGFLYDVKLVPDGKYGAQNDKGEWNGMVKELIDHRADLAVAPLTITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVRDGSTMTFFKKSKISTYEKMWAFMSSRQQSALVKNSDEGIQRVLTTDYALLMESTSIEYVTQRNCNLTQIGGLIDSKGYGVGTPIGSPYRDKITIAILQLQEEGKLHMMKEKWWRGNGCP 4dld B 2.0 BS01 TZG B 1 Y16 Y61 P88 L89 T90 R95 G140 S141 T142 S173 E190 S193 Y216 Y13 Y58 P85 L86 T87 R92 G137 S138 T139 S170 E187 S190 Y213 ? 0015276,0016020 Ki=1.5uM Ki=3000nM P22756 22407805 301 RTLIVTTILEEPYVMYRKSDKPLYGNDRFEGYCLDLLKELSNILGFLYDVKLVPDGKYGAQNDKGEWNGMVKELIDHRADLAVAPLTITYVREKVIDFSKPFMTLGISILYRKGTPIDSADDLAKQTKIEYGAVRDGSTMTFFKKSKISTYEKMWAFMSSRQQSALVKNSDEGIQRVLTTDYALLMESTSIEYVTQRNCNLTQIGGLIDSKGYGVGTPIGSPYRDKITIAILQLQEEGKLHMMKEKWWRGNGCP