1xap A 2.1 BS01 TTB A 1 F221 L224 L259 L262 F279 S280 R387 L407 F47 L50 L85 L88 F105 S106 R210 L230 ? 0003677,0004879,0005634,0006355,0048384 Kd=2.5nM -logKd/Ki=8.70, Kd=2nM EC50=4nM, Ki=0.500000nM, Kd=5nM, IC50=5nM P10826 15319780 1 AELDDLTEKIRKAHQETFPSLCQLGKYTTNSSADHRVRLDLGLWDKFSELATKCIIKIVEFAKRLPGFTGLTIADQITLLKAACLDILILRICTRYTPEQDTMTFSDGLTLNRTQMHNAGFGPLTDLVFTFANQLLPLEMDDTETGLLSAICLICGDRQDLEEPTKVDKLQEPLLEALKIYIRKRRPHMFPKILMKITDLRSISAKGAERVITLKMEIPGSMPPLIQEMLEN 4dm6 A 1.9 BS02 TTB A 1 F201 F230 L233 L271 I272 I275 F288 S289 F304 G393 R396 L416 F24 F53 L56 L94 I95 I98 F111 S112 F127 G216 R219 L239 ? 0003677,0004879,0005634,0006355,0048384 EC50=4nM, Ki=0.500000nM, Kd=5nM, IC50=5nM P10826 22355136 501 ESYEMTAELDDLTEKIRKAHQETFPSLCQLGKYTTNSSADHRVRLDLGLWDKFSELATKCIIKIVEFAKRLPGFTGLTIADQITLLKAACLDILILRICTRYTPEQDTMTFSDGLTLNRTQMHNAGFGPLTDLVFTFANQLLPLEMDDTETGLLSAICLICGDRQDLEEPTKVDKLQEPLLEALKIYIRKRRPSKPHMFPKILMKITDLRSISAKGAERVITLKMEIPGSMPPLIQEMLE 4dm6 B 1.9 BS02 TTB B 1 F1230 L1233 A1234 C1237 L1271 I1272 I1275 F1288 S1289 F1304 G1393 V1397 L1400 I1412 F51 L54 A55 C58 L92 I93 I96 F109 S110 F125 G214 V218 L221 I233 ? 0003677,0004879,0005634,0006355,0048384 EC50=4nM, Ki=0.500000nM, Kd=5nM, IC50=5nM P10826 22355136 1501 YEMTAELDDLTEKIRKAHQETFPSLCQLGKYTTNSSADHRVRLDLGLWDKFSELATKCIIKIVEFAKRLPGFTGLTIADQITLLKAACLDILILRICTRYTPEQDTMTFSDGLTLNRTQMHNAGFGPLTDLVFTFANQLLPLEMDDTETGLLSAICLICGDRQDLEEPTKVDKLQEPLLEALKIYIRKRRPSKPHMFPKILMKITDLRSISAKGAERVITLKMEIPGSMPPLIQEMLEN