3s68 A 1.85 BS02 TCW A 1 W38 W143 K144 N170 P174 E199 W36 W141 K142 N168 P172 E197 D141 K144 D169 N170 E199 D139 K142 D167 N168 E197 2.1.1.6 0000287,0006584,0008171,0016206 -logKd/Ki=8.66, IC50=2.2nM IC50=2.2nM P22734 22349227 227 DTKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEMNPDYAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEKCGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGP 4d7b A 1.15 BS01 TCW B 1 K15 L17 A108 L110 S117 K6 L8 A99 L101 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=21nM -logKd/Ki=7.68, Kd=21nM Kd=56nM P02766 26902880 1126 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 4d7b B 1.15 BS01 TCW A 1 K15 L17 A108 S117 K6 L8 A99 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=21nM -logKd/Ki=7.68, Kd=21nM Kd=56nM P02766 26902880 1126 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 4pyl A 2.2 BS03 TCW A 1 W81 M83 D184 W186 K187 N213 P217 E242 W35 M37 D138 W140 K141 N167 P171 E196 D184 K187 D212 N213 E242 D138 K141 D166 N167 E196 2.1.1.6 0000287,0006584,0008171,0016206 IC50=2.2nM P22734 25084335 303 TKEQRILRYVQQNAKPGDPQSVLEAIDTYCTQKEWAMNVGDAKGQIMDAVIREYSPSLVLELGAYCGYSAVRMARLLQPGARLLTMEMNPDYAAITQQMLNFAGLQDKVTILNGASQDLIPQLKKKYDVDTLDMVFLDHWKDRYLPDTLLLEKCGLLRKGTVLLADNVIVPGTPDFLAYVRGSSSFECTHYSSYLEYMKVVDGLEKAIYQGPS 5a6i A 1.86 BS01 TCW A 1 K15 L17 A108 S117 T118 K6 L8 A99 S108 T109 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=56nM -logKd/Ki=7.25, Kd=56nM Kd=56nM P02766 26902880 1124 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVIT 6txv A 1.6 BS01 TCW A 1 K15 L17 A108 L110 S117 K6 L8 A99 L101 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=3.1uM Kd=56nM P02766 32324953 201 CPLMVKVLDAVRGSPTINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 6txv B 1.6 BS01 TCW B 1 K15 L17 A108 L110 S117 K6 L8 A99 L101 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=3.1uM Kd=56nM P02766 32324953 201 CPLMVKVLDAVRGSPTINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 6txw A 1.153 BS01 TCW A 1 K15 L17 A108 L110 S117 K6 L8 A99 L101 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=0.11uM Kd=56nM P02766 32324953 201 CPLMVKVLDAVRGSPAINVAGHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 6txw B 1.153 BS01 TCW B 1 K15 L17 A108 L110 S117 K6 L8 A99 L101 S108 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=0.11uM Kd=56nM P02766 32324953 201 CPLMVKVLDAVRGSPAINVAGHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 6xtk A 1.7 BS01 TCW A 1 K15 L17 A108 S117 T118 K6 L8 A99 S108 T109 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=0.029uM Kd=56nM P02766 32324953 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPCSYSTTAVVTNP 6xtk B 1.7 BS01 TCW B 1 K15 L17 A108 S117 T118 K6 L8 A95 S104 T105 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 Kd=0.029uM Kd=56nM P02766 32324953 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANRRYTIAALLSPCSYSTTAVVTNP 7ybr A 1.71 BS01 TCW A 1 K15 L17 A108 S117 T118 K6 L8 A96 S105 T106 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 P02766 36851846 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTSNDRRYTIAALLSPYSYSTTAVVTN 7ybr B 1.71 BS01 TCW B 1 K15 L17 A108 S117 T118 K6 L8 A99 S108 T109 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 P02766 36851846 201 CPLMVKVLDAVRGSPAINVAVHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTSNDSGPRRYTIAALLSPYSYSTTAVVTN 8guv A 1.32 BS02 TCW A 1 Y36 H50 D100 V101 T104 N107 Y36 H50 D100 V101 T104 N107 ? 0005737,0007157,0009986,0030246,0042597 Q05097 302 AWKGEVLANNEAGQVTSIIYNPGDVITIVAAGWASYGPTQKWGPQGDREHPDQGLICHDAFCGALVMKIGNSGTIPVNTGLFRWVAPNNVQGAITLIYNDVPGTYGNNSGSFSVNIGKDQS 8guv B 1.32 BS02 TCW B 1 Y36 H50 D100 T104 N107 Y36 H50 D100 T104 N107 ? 0005737,0007157,0009986,0030246,0042597 Q05097 302 AWKGEVLANNEAGQVTSIIYNPGDVITIVAAGWASYGPTQKWGPQGDREHPDQGLICHDAFCGALVMKIGNSGTIPVNTGLFRWVAPNNVQGAITLIYNDVPGTYGNNSGSFSVNIGKDQS 8guv B 1.32 BS03 TCW B 2 Y36 G37 H50 P51 Y36 G37 H50 P51 ? 0005737,0007157,0009986,0030246,0042597 Q05097 303 AWKGEVLANNEAGQVTSIIYNPGDVITIVAAGWASYGPTQKWGPQGDREHPDQGLICHDAFCGALVMKIGNSGTIPVNTGLFRWVAPNNVQGAITLIYNDVPGTYGNNSGSFSVNIGKDQS 8pm8 A 1.57 BS01 TCW A 1 K15 L17 A108 L110 S117 T118 T119 K6 L8 A99 L101 S108 T109 T110 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 P02766 37837673 201 CPLMVKVLDAVRGSPAINVAMHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP 8pm8 B 1.57 BS01 TCW B 1 K15 L17 A108 L110 S117 T118 T119 K6 L8 A99 L101 S108 T109 T110 ? 0005179,0005515,0005576,0005615,0005737,0006144,0007165,0035578,0042802,0070062,0070324 P02766 37837673 201 CPLMVKVLDAVRGSPAINVAMHVFRKAADDTWEPFASGKTSESGELHGLTTEEEFVEGIYKVEIDTKSYWKALGISPFHEHAEVVFTANDSGPRRYTIAALLSPYSYSTTAVVTNP