2x22 A 2.1 BS02 TCU A 1 G96 F97 F149 Y158 M161 A198 I202 V203 G95 F96 F148 Y157 M160 A197 I201 V202 Y158 K165 Y157 K164 1.3.1.9 0004318,0005504,0005886,0006633,0009274,0016491,0030497,0046677,0050343,0070403,0071768 Ki=7.8nM Ki=913nM, IC50=51nM P9WGR1 20200152 1271 TGLLDGKRILVSGIITDSSIAFHIARVAQEQGAQLVLTGFDRLRLIQRITDRLPAKAPLLELDVQNEEHLASLAGRVTEAIGAGNKLDGVVHSIGFMPQTGMGINPFFDAPYADVSKGIHISAYSYASMAKALLPIMNPGGSIVGMDFDPSRAMPAYNWMTVAKSALESVNRFVAREAGKYGVRSNLVAAGPIRTLAMSAIVGGALGEEAGAQIQLLEEGWDQRAPIGWNMKDATPVAKTVCALLSDWLPATTGDIIYADGGAHTQLL 2x22 B 2.1 BS02 TCU B 1 G96 F149 A157 Y158 M161 V203 G95 F148 A156 Y157 M160 V202 Y158 K165 Y157 K164 1.3.1.9 0004318,0005504,0005886,0006633,0009274,0016491,0030497,0046677,0050343,0070403,0071768 Ki=7.8nM Ki=913nM, IC50=51nM P9WGR1 20200152 1271 TGLLDGKRILVSGIITDSSIAFHIARVAQEQGAQLVLTGFDRLRLIQRITDRLPAKAPLLELDVQNEEHLASLAGRVTEAIGAGNKLDGVVHSIGFMPQTGMGINPFFDAPYADVSKGIHISAYSYASMAKALLPIMNPGGSIVGMDFDPSRAMPAYNWMTVAKSALESVNRFVAREAGKYGVRSNLVAAGPIRTLAMSAIVGGALGEEAGAQIQLLEEGWDQRAPIGWNMKDATPVAKTVCALLSDWLPATTGDIIYADGGAHTQLL 2x23 A 1.807 BS02 TCU A 1 G96 F97 F149 Y158 M161 A198 I202 V203 G95 F96 F148 Y157 M160 A197 I201 V202 Y158 K165 Y157 K164 1.3.1.9 0004318,0005504,0005886,0006633,0009274,0016491,0030497,0046677,0050343,0070403,0071768 Ki=7.8nM Ki=913nM, IC50=51nM P9WGR1 20200152 1271 TGLLDGKRILVSGIITDSSIAFHIARVAQEQGAQLVLTGFDRLRLIQRITDRLPAKAPLLELDVQNEEHLASLAGRVTEAIGAGNKLDGVVHSIGFMPQTGMGINPFFDAPYADVSKGIHISAYSYASMAKALLPIMNPGGSIVGMDFDPSRAMPAYNWMTVAKSALESVNRFVAREAGKYGVRSNLVAAGPIRTLAMSAIVGGALGEEAGAQIQLLEEGWDQRAPIGWNMKDATPVAKTVCALLSDWLPATTGDIIYADGGAHTQLL 2x23 B 1.807 BS02 TCU B 1 G96 F97 F149 Y158 M161 A198 M199 I202 G95 F96 F148 Y157 M160 A197 M198 I201 Y158 K165 Y157 K164 1.3.1.9 0004318,0005504,0005886,0006633,0009274,0016491,0030497,0046677,0050343,0070403,0071768 Ki=7.8nM Ki=913nM, IC50=51nM P9WGR1 20200152 1271 TGLLDGKRILVSGIITDSSIAFHIARVAQEQGAQLVLTGFDRLRLIQRITDRLPAKAPLLELDVQNEEHLASLAGRVTEAIGAGNKLDGVVHSIGFMPQTGMGINPFFDAPYADVSKGIHISAYSYASMAKALLPIMNPGGSIVGMDFDPSRAMPAYNWMTVAKSALESVNRFVAREAGKYGVRSNLVAAGPIRTLAMSAIVGGALGEEAGAQIQLLEEGWDQRAPIGWNMKDATPVAKTVCALLSDWLPATTGDIIYADGGAHTQLL 2x23 E 1.807 BS02 TCU E 1 G96 F97 F149 Y158 M161 A198 I202 G95 F96 F148 Y157 M160 A197 I201 1.3.1.9 0004318,0005504,0005886,0006633,0009274,0016491,0030497,0046677,0050343,0070403,0071768 Ki=7.8nM Ki=913nM, IC50=51nM P9WGR1 20200152 1271 TGLLDGKRILVSGIITDSSIAFHIARVAQEQGAQLVLTGFDRLRLIQRITDRLPAKAPLLELDVQNEEHLASLAGRVTEAIGAGNKLDGVVHSIGFMPQTGMGINPFFDAPYADVSKGIHISAYSYASMAKALLPIMNPGGSIVGMDFDPSRAMPAYNWMTVAKSALESVNRFVAREAGKYGVRSNLVAAGPIRTLAMSAIVGGALGEEAGAQIQLLEEGWDQRAPIGWNMKDATPVAKTVCALLSDWLPATTGDIIYADGGAHTQLL 2x23 G 1.807 BS02 TCU G 1 G96 F97 F149 Y158 M161 A198 M199 I202 G95 F96 F148 Y157 M160 A197 M198 I201 1.3.1.9 0004318,0005504,0005886,0006633,0009274,0016491,0030497,0046677,0050343,0070403,0071768 Ki=7.8nM Ki=913nM, IC50=51nM P9WGR1 20200152 1271 TGLLDGKRILVSGIITDSSIAFHIARVAQEQGAQLVLTGFDRLRLIQRITDRLPAKAPLLELDVQNEEHLASLAGRVTEAIGAGNKLDGVVHSIGFMPQTGMGINPFFDAPYADVSKGIHISAYSYASMAKALLPIMNPGGSIVGMDFDPSRAMPAYNWMTVAKSALESVNRFVAREAGKYGVRSNLVAAGPIRTLAMSAIVGGALGEEAGAQIQLLEEGWDQRAPIGWNMKDATPVAKTVCALLSDWLPATTGDIIYADGGAHTQLL 4bnm A 2.35 BS01 TCU A 1 A95 Y147 Y157 S197 A198 V201 I207 A93 Y145 Y155 S195 A196 V199 I205 Y147 Y157 M160 K164 K199 Y145 Y155 M158 K162 K197 1.3.1.39 0000166,0004318,0006633,0016491,0042802,0141148 A0A0H3JLH9 23697754 1257 NLENKTYVIMGIANKRSIAFGVAKVLDQLGAKLVFTYRKERSRKELEKLLEQLNQPEAHLYQIDVQSDEEVINGFEQIGKDVGNIDGVYHSIAFANMEDLRGRFSETSREGFLLAQDISSYSLTIVAHEAKKLMPEGGSIVATTYLGGEFAVQNYNVMGVAKASLEANVKYLALDLGPDNIRVNAISAGPIRTLSAKGVGGFNTILKEIEERAPLKRNVDQVEVGKTAAYLLSDLSSGVTGENIHVDSGFHAIK 4bnm B 2.35 BS03 TCU B 1 A95 Y147 Y157 M160 S197 A198 V201 A94 Y146 Y156 M159 S196 A197 V200 Y147 Y157 M160 K164 K199 Y146 Y156 M159 K163 K198 1.3.1.39 0000166,0004318,0006633,0016491,0042802,0141148 A0A0H3JLH9 23697754 1258 VNLENKTYVIMGIANKRSIAFGVAKVLDQLGAKLVFTYRKERSRKELEKLLEQLNQPEAHLYQIDVQSDEEVINGFEQIGKDVGNIDGVYHSIAFANMEDLRGRFSETSREGFLLAQDISSYSLTIVAHEAKKLMPEGGSIVATTYLGGEFAVQNYNVMGVAKASLEANVKYLALDLGPDNIRVNAISAGPIRTLSAKGVGGFNTILKEIEERAPLKRNVDQVEVGKTAAYLLSDLSSGVTGENIHVDSGFHAIK 4bnm C 2.35 BS02 TCU C 1 A95 Y147 Y157 M160 S197 V201 A94 Y146 Y156 M159 S196 V200 Y147 Y157 M160 K164 K199 Y146 Y156 M159 K163 K198 1.3.1.39 0000166,0004318,0006633,0016491,0042802,0141148 A0A0H3JLH9 23697754 1258 VNLENKTYVIMGIANKRSIAFGVAKVLDQLGAKLVFTYRKERSRKELEKLLEQLNQPEAHLYQIDVQSDEEVINGFEQIGKDVGNIDGVYHSIAFANMEDLRGRFSETSREGFLLAQDISSYSLTIVAHEAKKLMPEGGSIVATTYLGGEFAVQNYNVMGVAKASLEANVKYLALDLGPDNIRVNAISAGPIRTLSAKGVGGFNTILKEIEERAPLKRNVDQVEVGKTAAYLLSDLSSGVTGENIHVDSGFHAIK 4bnm D 2.35 BS02 TCU D 1 A95 Y147 Y157 S197 V201 F204 A93 Y145 Y155 S195 V199 F202 Y147 Y157 M160 K164 K199 Y145 Y155 M158 K162 K197 1.3.1.39 0000166,0004318,0006633,0016491,0042802,0141148 A0A0H3JLH9 23697754 1258 NLENKTYVIMGIANKRSIAFGVAKVLDQLGAKLVFTYRKERSRKELEKLLEQLNQPEAHLYQIDVQSDEEVINGFEQIGKDVGNIDGVYHSIAFANMEDLRGRFSETSREGFLLAQDISSYSLTIVAHEAKKLMPEGGSIVATTYLGGEFAVQNYNVMGVAKASLEANVKYLALDLGPDNIRVNAISAGPIRTLSAKGVGGFNTILKEIEERAPLKRNVDQVEVGKTAAYLLSDLSSGVTGENIHVDSGFHAIK 4bnm E 2.35 BS02 TCU E 1 Y147 Y157 S197 Y146 Y156 S196 Y147 Y157 M160 K164 K199 Y146 Y156 M159 K163 K198 1.3.1.39 0000166,0004318,0006633,0016491,0042802,0141148 A0A0H3JLH9 23697754 1258 VNLENKTYVIMGIANKRSIAFGVAKVLDQLGAKLVFTYRKERSRKELEKLLEQLNQPEAHLYQIDVQSDEEVINGFEQIGKDVGNIDGVYHSIAFANMEDLRGRFSETSREGFLLAQDISSYSLTIVAHEAKKLMPEGGSIVATTYLGGEFAVQNYNVMGVAKASLEANVKYLALDLGPDNIRVNAISAGPIRTLSAKGVGGFNTILKEIEERAPLKRNVDQVEVGKTAAYLLSDLSSGVTGENIHVDSGFHAIK 4bnm F 2.35 BS03 TCU F 1 A95 Y157 M160 S197 V201 A94 Y156 M159 S196 V200 Y147 Y157 M160 K164 K199 Y146 Y156 M159 K163 K198 1.3.1.39 0000166,0004318,0006633,0016491,0042802,0141148 A0A0H3JLH9 23697754 1258 VNLENKTYVIMGIANKRSIAFGVAKVLDQLGAKLVFTYRKERSRKELEKLLEQLNQPEAHLYQIDVQSDEEVINGFEQIGKDVGNIDGVYHSIAFANMEDLRGRFSETSREGFLLAQDISSYSLTIVAHEAKKLMPEGGSIVATTYLGGEFAVQNYNVMGVAKASLEANVKYLALDLGPDNIRVNAISAGPIRTLSAKGVGGFNTILKEIEERAPLKRNVDQVEVGKTAAYLLSDLSSGVTGENIHVDSGFHAIK 4bnm G 2.35 BS03 TCU G 1 A95 Y147 Y157 M160 S197 V201 A94 Y146 Y156 M159 S196 V200 Y147 Y157 M160 K164 K199 Y146 Y156 M159 K163 K198 1.3.1.39 0000166,0004318,0006633,0016491,0042802,0141148 A0A0H3JLH9 23697754 1258 VNLENKTYVIMGIANKRSIAFGVAKVLDQLGAKLVFTYRKERSRKELEKLLEQLNQPEAHLYQIDVQSDEEVINGFEQIGKDVGNIDGVYHSIAFANMEDLRGRFSETSREGFLLAQDISSYSLTIVAHEAKKLMPEGGSIVATTYLGGEFAVQNYNVMGVAKASLEANVKYLALDLGPDNIRVNAISAGPIRTLSAKGVGGFNTILKEIEERAPLKRNVDQVEVGKTAAYLLSDLSSGVTGENIHVDSGFHAIK 4bnm H 2.35 BS02 TCU H 1 Y147 Y157 S197 A198 V201 I207 Y145 Y155 S195 A196 V199 I205 Y147 Y157 M160 K164 K199 Y145 Y155 M158 K162 K197 1.3.1.39 0000166,0004318,0006633,0016491,0042802,0141148 A0A0H3JLH9 23697754 1258 NLENKTYVIMGIANKRSIAFGVAKVLDQLGAKLVFTYRKERSRKELEKLLEQLNQPEAHLYQIDVQSDEEVINGFEQIGKDVGNIDGVYHSIAFANMEDLRGRFSETSREGFLLAQDISSYSLTIVAHEAKKLMPEGGSIVATTYLGGEFAVQNYNVMGVAKASLEANVKYLALDLGPDNIRVNAISAGPIRTLSAKGVGGFNTILKEIEERAPLKRNVDQVEVGKTAAYLLSDLSSGVTGENIHVDSGFHAIK 5coq A 2.3 BS02 TCU A 1 G96 F97 M103 F149 Y158 M161 A198 M199 G95 F96 M102 F148 Y157 M160 A197 M198 Y158 K165 Y157 K164 1.3.1.9 0004318,0005504,0005886,0006633,0009274,0016491,0030497,0046677,0050343,0070403,0071768 Ki=427.5nM Ki=913nM, IC50=51nM P9WGR1 26147157 301 TGLLDGKRILVSGIITDSSIAFHIARVAQEQGAQLVLTGFDRLRLIQRITDRLPAKAPLLELDVQNEEHLASLAGRVTEAIGAGNKLDGVVHSIGFMPQTGMGINPFFDAPYADVSKGIHISAYSYASMAKALLPIMNPGGSIVGMDFDPSRAMPAYNWMTVAKSALESVNRFVAREAGKYGVRSNLVAAGPIRTLAMSAIAGGEAGAQIQLLEEGWDQRAPIGWNMKDATPVAKTVCALLSDWLPATTGDIIYADGGAHTQLL 5coq B 2.3 BS02 TCU B 1 G96 F97 F149 Y158 A198 M199 G95 F96 F148 Y157 A197 M198 Y158 K165 Y157 K164 1.3.1.9 0004318,0005504,0005886,0006633,0009274,0016491,0030497,0046677,0050343,0070403,0071768 Ki=427.5nM Ki=913nM, IC50=51nM P9WGR1 26147157 301 TGLLDGKRILVSGIITDSSIAFHIARVAQEQGAQLVLTGFDRLRLIQRITDRLPAKAPLLELDVQNEEHLASLAGRVTEAIGAGNKLDGVVHSIGFMPQTGMGINPFFDAPYADVSKGIHISAYSYASMAKALLPIMNPGGSIVGMDFDPSRAMPAYNWMTVAKSALESVNRFVAREAGKYGVRSNLVAAGPIRTLAMSAIAGGALGEEAGAQIQLLEEGWDQRAPIGWNMKDATPVAKTVCALLSDWLPATTGDIIYADGGAHTQLL 5coq C 2.3 BS02 TCU C 1 G96 F97 M103 F149 Y158 M161 A198 G95 F96 M102 F148 Y157 M160 A197 Y158 K165 Y157 K164 1.3.1.9 0004318,0005504,0005886,0006633,0009274,0016491,0030497,0046677,0050343,0070403,0071768 Ki=427.5nM Ki=913nM, IC50=51nM P9WGR1 26147157 302 TGLLDGKRILVSGIITDSSIAFHIARVAQEQGAQLVLTGFDRLRLIQRITDRLPAKAPLLELDVQNEEHLASLAGRVTEAIGAGNKLDGVVHSIGFMPQTGMGINPFFDAPYADVSKGIHISAYSYASMAKALLPIMNPGGSIVGMDFDPSRAMPAYNWMTVAKSALESVNRFVAREAGKYGVRSNLVAAGPIRTLAMSAIAQIQLLEEGWDQRAPIGWNMKDATPVAKTVCALLSDWLPATTGDIIYADGGAHTQLL 5coq D 2.3 BS02 TCU D 1 G96 F97 M103 F149 Y158 M161 A198 M199 I202 I215 G95 F96 M102 F148 Y157 M160 A197 M198 I201 I208 Y158 K165 Y157 K164 1.3.1.9 0004318,0005504,0005886,0006633,0009274,0016491,0030497,0046677,0050343,0070403,0071768 Ki=427.5nM Ki=913nM, IC50=51nM P9WGR1 26147157 301 TGLLDGKRILVSGIITDSSIAFHIARVAQEQGAQLVLTGFDRLRLIQRITDRLPAKAPLLELDVQNEEHLASLAGRVTEAIGAGNKLDGVVHSIGFMPQTGMGINPFFDAPYADVSKGIHISAYSYASMAKALLPIMNPGGSIVGMDFDPSRAMPAYNWMTVAKSALESVNRFVAREAGKYGVRSNLVAAGPIRTLAMSAIAEAGAQIQLLEEGWDQRAPIGWNMKDATPVAKTVCALLSDWLPATTGDIIYADGGAHTQLL 5cp8 A 2.4 BS02 TCU A 1 G96 F97 M103 F149 Y158 A198 M199 A215 G94 F95 M101 F147 Y156 A196 M197 A213 Y158 K165 Y156 K163 1.3.1.9 0004318,0005504,0005886,0006633,0009274,0016491,0030497,0046677,0050343,0070403,0071768 Ki=1570.6nM Ki=913nM, IC50=51nM P9WGR1 26147157 301 GLLDGKRILVSGIITDSSIAFHIARVAQEQGAQLVLTGFDRLRLIQRITDRLPAKAPLLELDVQNEEHLASLAGRVTEAIGAGNKLDGVVHSIGFMPQTGMGINPFFDAPYADVSKGIHISAYSYASMAKALLPIMNPGGSIVGMDFDPSRAMPAYNWMTVAKSALESVNRFVAREAGKYGVRSNLVAAGPIRTLAMSAIVGGALGEEAGAQAQLLEEGWDQRAPIGWNMKDATPVAKTVCALLSDWLPATTGDIIYADGGAHTQLL