4xry	A	2.5	BS02	SI5	A	1	F120 E216 Q244 S304 A305 F483	F87 E183 Q211 S271 A272 F450	T309 F436 C443	T276 F403 C410	1.14.14.-	0004497,0005506,0005737,0005739,0005783,0005789,0006631,0006805,0008202,0008203,0008210,0009804,0009820,0009822,0016020,0016098,0016491,0016705,0016712,0019369,0020037,0033076,0042178,0042572,0042759,0043231,0046872,0051100,0062187,0062188,0062189,0070989,0090350		ic50=13.9uM		IC50=13900nM	P10635	25781223	602 	GKLPPGPLPLPGLGNLLHVDTPYCFDQLRRRFGDVFSLQLAWTPVVVLNGLAAVREALVTHGEDTADRPPVPITQILGFGPRSQGVFLARYGPAWREQRRFSVSTLRNLGLGKKSLEQWVTEEAACLCAAFANHSGRPFRPNGLLDKAVSNVIASLTCGRRFEYDDPRFLRLLDLAQEGLKEESGFLREVLNAVPVLLHIPALAGKVLRFQKAFLTQLDELLTEHRMTWDPAQPPRDLTEAFLAEMEKAKGNPESSFNDENLRIVVADLFSAGMVTTSTTLAWGLLLMILHPDVQRRVQQEIDDVIGQVRRPEMGDQAHMPYTTAVIHEVQRFGDIVPLGVTHMTSRDIEVQGFRIPKGTTLITNLSSVLKDEAVWEKPFRFHPEHFLDAQGHFVKPEAFLPFSAGRRACLGEPLARMELFLFFTSLLQHFSFSVPTGQPRPSHHGVFAFLVSPSPYELCAVPR
4xry	B	2.5	BS03	SI5	B	1	F120 G212 E216 D301 S304 A305 F483 L484	F82 G170 E174 D259 S262 A263 F441 L442	T309 F436 C443	T267 F394 C401	1.14.14.-	0004497,0005506,0005737,0005739,0005783,0005789,0006631,0006805,0008202,0008203,0008210,0009804,0009820,0009822,0016020,0016098,0016491,0016705,0016712,0019369,0020037,0033076,0042178,0042572,0042759,0043231,0046872,0051100,0062187,0062188,0062189,0070989,0090350		ic50=13.9uM		IC50=13900nM	P10635	25781223	602 	GKLPPGPLPGNLLHVTPYCFDQLRRRFGDVFSLQLAWTPVVVLNGLAAVREALVTHGEDTADRPPVPITQILGFGPRSQGVFLARYGPAWREQRRFSVSTLRNLKSLEQWVTEEAACLCAAFANHSGRPFRPNGLLDKAVSNVIASLTCGRRFEYDDPRFLRLLDLAQEGLKEESGFLREVLNAVPVLLHIPALAGKVLRFQKAFLTQLDELLTEHRMTWDPAQPPRDLTEAFLAEMEKAKGNPESSFNDENLRIVVADLFSAGMVTTSTTLAWGLLLMILHPDVQRRVQQEIDDVIGQVRRPEMGDQAHMPYTTAVIHEVQRFGDIVPLGVTHMTSRDIEVQGFRIPKGTTLITNLSSVLKDEAVWEKPFRFHPEHFLDAQGHFVKPEAFLPFSAGRRACLGEPLARMELFLFFTSLLQHFSFSVPTGQPRPSHHGVFAFLVSPSPYELCAVPR
4xry	C	2.5	BS02	SI5	C	1	F120 G212 E216 Q244 S304 A305 T309 F483 L484	F74 G161 E165 Q193 S253 A254 T258 F432 L433	T309 F436 C443	T258 F385 C392	1.14.14.-	0004497,0005506,0005737,0005739,0005783,0005789,0006631,0006805,0008202,0008203,0008210,0009804,0009820,0009822,0016020,0016098,0016491,0016705,0016712,0019369,0020037,0033076,0042178,0042572,0042759,0043231,0046872,0051100,0062187,0062188,0062189,0070989,0090350		ic50=13.9uM		IC50=13900nM	P10635	25781223	602 	LPPGPLPTPYCFDQLRRRFGDVFSLQLAWTPVVVLNGLAAVREALVTHGEDTADRPPVPITQILGFGPRSQGVFLARYGPAWREQRRFSVSTLRNLSLEQWVTEEAACLCAAFANHSGRPFRPNGLLDKAVSNVIASLTCGRRFEYDDPRFLRLLDLAQEGLKEESGFLREVLNAVPVLLHIPALAGKVLRFQKAFLTQLDELLTEHRMTWDPAQPPRDLTEAFLAEMEKAKGNPESSFNDENLRIVVADLFSAGMVTTSTTLAWGLLLMILHPDVQRRVQQEIDDVIGQVRRPEMGDQAHMPYTTAVIHEVQRFGDIVPLGVTHMTSRDIEVQGFRIPKGTTLITNLSSVLKDEAVWEKPFRFHPEHFLDAQGHFVKPEAFLPFSAGRRACLGEPLARMELFLFFTSLLQHFSFSVPTGQPRPSHHGVFAFLVSPSPYELCAVPR
4xry	D	2.5	BS02	SI5	D	1	F120 E216 Q244 S304 A305 F483	F75 E171 Q199 S259 A260 F438	T309 F436 C443	T264 F391 C398	1.14.14.-	0004497,0005506,0005737,0005739,0005783,0005789,0006631,0006805,0008202,0008203,0008210,0009804,0009820,0009822,0016020,0016098,0016491,0016705,0016712,0019369,0020037,0033076,0042178,0042572,0042759,0043231,0046872,0051100,0062187,0062188,0062189,0070989,0090350		ic50=13.9uM		IC50=13900nM	P10635	25781223	602 	LPPGPLPLTPYCFDQLRRRFGDVFSLQLAWTPVVVLNGLAAVREALVTHGEDTADRPPVPITQILGFGPRSQGVFLARYGPAWREQRRFSVSTLRNLGLGKKSLEQWVTEEAACLCAAFANHSGRPFRPNGLLDKAVSNVIASLTCGRRFEYDDPRFLRLLDLAQEGLKEESGFLREVLNAVPVLLHIPALAGKVLRFQKAFLTQLDELLTEHRMTWDPAQPPRDLTEAFLAEMEKAKGNPESSFNDENLRIVVADLFSAGMVTTSTTLAWGLLLMILHPDVQRRVQQEIDDVIGQVRRPEMGDQAHMPYTTAVIHEVQRFGDIVPLGVTHMTSRDIEVQGFRIPKGTTLITNLSSVLKDEAVWEKPFRFHPEHFLDAQGHFVKPEAFLPFSAGRRACLGEPLARMELFLFFTSLLQHFSFSVPTGQPRPSHHGVFAFLVSPSPYELCAVPR
4xxs	A	1.86	BS01	SI5	A	1	D32 G34 S35 Y71 F108 W115 R128 D228 G230	D37 G39 S40 Y76 F113 W120 R133 D224 G226	D32 S35 N37 A39 Y71 D228 T231	D37 S40 N42 A44 Y76 D224 T227	3.4.23.46	0004190,0006508,0016020		ic50=52nM	-logKd/Ki=7.28, IC50=52nM	IC50=4.0nM	P56817	25781223	401 	RGSFVEMVDNLRGKSGQGYYVEMTVGSPPQTLNILVDTGSSNFAVGAAPHPFLHRYYQRQLSSTYRDLRKGVYVPYTQGKWEGELGTDLVSIPHGPNVTVRANIAAITESDKFFINGSNWEGILGLAYAEIARPDDSLEPFFDSLVKQTHVPNLFSLQLCGALASVGGSMIIGGIDHSLYTGSLWYTPIRREWYYEVIIVRVEINGQDLKMDCKEYNYDKSIVDSGTTNLRLPKKVFEAAVKSIKAASSTEKFPDGFWLGEQLVCWQAGTTPWNIFPVISLYLMGEVTNQSFRITILPQQYLRPVDDCYKFAISQSSTGTVMGAVIMEGFYVVFDRARKRIGFAVSACHVHDEFRTAAVEGPFVTLDMEDCGYNIP