1hv5 A 2.6 BS04 RXP A 1 L172 G179 I180 L181 A182 A184 Q215 H219 E220 F240 Y241 L72 G79 I80 L81 A82 A84 Q115 H119 E120 F140 Y141 H219 E220 H223 H229 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 -logKd/Ki=8.30, Ki=5nM Ki=5nM Q02853 11254383 6001 MFVLSGGRWEKTDLTYRILRFPWQLVREQVRQTVAEALQVWSEVTPLTFTEVHEGRADIMIDFARYWHGDNLPFDGPGGILAHAFFPKTHREGDVHFDYDETWTIGDNQGTDLLQVAAHEFGHVLGLQHTTAAKALMSPFYTFRYPLSLSPDDRRGIQHLYG 1hv5 B 2.6 BS04 RXP B 1 L172 G179 I180 L181 A182 A184 Q215 H219 E220 H223 F240 Y241 L72 G79 I80 L81 A82 A84 Q115 H119 E120 H123 F140 Y141 H219 E220 H223 H229 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 Ki=5nM Q02853 11254383 6002 MFVLSGGRWEKTDLTYRILRFPWQLVREQVRQTVAEALQVWSEVTPLTFTEVHEGRADIMIDFARYWHGDNLPFDGPGGILAHAFFPKTHREGDVHFDYDETWTIGDNQGTDLLQVAAHEFGHVLGLQHTTAAKALMSPFYTFRYPLSLSPDDRRGIQHLYGRP 1hv5 C 2.6 BS04 RXP C 1 G179 I180 L181 A182 H183 A184 Q215 H219 E220 H223 H229 F240 Y241 G79 I80 L81 A82 H83 A84 Q115 H119 E120 H123 H129 F140 Y141 H219 E220 H223 H229 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 Ki=5nM Q02853 11254383 6003 MFVLSGGRWEKTDLTYRILRFPWQLVREQVRQTVAEALQVWSEVTPLTFTEVHEGRADIMIDFARYWHGDNLPFDGPGGILAHAFFPKTHREGDVHFDYDETWTIGDNQGTDLLQVAAHEFGHVLGLQHTTAAKALMSPFYTFRYPLSLSPDDRRGIQHLYG 1hv5 D 2.6 BS04 RXP D 1 G179 I180 L181 A182 A184 Q215 H219 E220 H229 L236 F240 Y241 G79 I80 L81 A82 A84 Q115 H119 E120 H129 L136 F140 Y141 H219 E220 H223 H229 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 Ki=5nM Q02853 11254383 6004 MFVLSGGRWEKTDLTYRILRFPWQLVREQVRQTVAEALQVWSEVTPLTFTEVHEGRADIMIDFARYWHGDNLPFDGPGGILAHAFFPKTHREGDVHFDYDETWTIGDNQGTDLLQVAAHEFGHVLGLQHTTAAKALMSPFYTFRYPLSLSPDDRRGIQHLYG 1hv5 E 2.6 BS04 RXP E 1 I180 L181 A182 A184 Q215 H219 E220 H223 S238 F240 Y241 I80 L81 A82 A84 Q115 H119 E120 H123 S138 F140 Y141 H219 E220 H223 H229 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 Ki=5nM Q02853 11254383 6005 MFVLSGGRWEKTDLTYRILRFPWQLVREQVRQTVAEALQVWSEVTPLTFTEVHEGRADIMIDFARYWHGDNLPFDGPGGILAHAFFPKTHREGDVHFDYDETWTIGDNQGTDLLQVAAHEFGHVLGLQHTTAAKALMSPFYTFRYPLSLSPDDRRGIQHLYGRPQ 1hv5 F 2.6 BS04 RXP F 1 L172 G179 I180 L181 A182 A184 H219 E220 H229 F240 Y241 L72 G79 I80 L81 A82 A84 H119 E120 H129 F140 Y141 H219 E220 H223 H229 H119 E120 H123 H129 3.4.24.- 0004222,0006508,0008237,0008270,0031012 Ki=5nM Q02853 11254383 6006 MFVLSGGRWEKTDLTYRILRFPWQLVREQVRQTVAEALQVWSEVTPLTFTEVHEGRADIMIDFARYWHGDNLPFDGPGGILAHAFFPKTHREGDVHFDYDETWTIGDNQGTDLLQVAAHEFGHVLGLQHTTAAKALMSPFYTFRYPLSLSPDDRRGIQHLYG