1c9h A 2.0 BS01 RAP A 1 Y26 F36 D37 F46 Q53 E54 V55 I56 F59 Y82 H87 Y26 F36 D37 F46 Q53 E54 V55 I56 F59 Y82 H87 Y26 F36 D37 I56 Y82 F99 Y26 F36 D37 I56 Y82 F99 5.2.1.8 0002027,0003755,0005102,0005219,0005515,0005528,0005737,0006458,0006939,0007204,0009749,0010459,0010880,0010881,0016020,0016247,0016529,0019227,0019722,0019855,0022417,0030018,0030073,0030551,0033017,0033197,0034704,0035773,0042026,0042098,0042542,0044325,0048680,0050849,0051209,0051280,0051284,0051775,0060314,0061179 Kd=0.200000nM P68106 10713512 108 GVEIETISPGDGRTFPKKGQTCVVHYTGMLQNGKKFDSSRDRNKPFKFRIGKQEVIKGFEEGAAQMSLGQRAKLTCTPDVAYGATGHPGVIPPNATLIFDVELLNLE 1fap A 2.7 BS01 RAP A 1 F36 D37 F46 Q53 E54 V55 I56 W59 Y82 F36 D37 F46 Q53 E54 V55 I56 W59 Y82 Y26 F36 D37 I56 Y82 F99 Y26 F36 D37 I56 Y82 F99 5.2.1.8 0000413,0003007,0003755,0005160,0005515,0005527,0005528,0005737,0005829,0006457,0006458,0014802,0014809,0016020,0016247,0016529,0022417,0030018,0030512,0030547,0032092,0032880,0032926,0033017,0034713,0042026,0042110,0043123,0044325,0050776,0055010,0060314,0060347,0070411,0070588,0070697,0097435,0098562,1902991,1990000,1990425 IC50=0.600000nM, EC50=30nM, Ki=0.20nM P62942 8662507 108 GVQVETISPGDGRTFPKRGQTCVVHYTGMLEDGKKFDSSRDRNKPFKFMLGKQEVIRGWEEGVAQMSVGQRAKLTISPDYAYGATGHPGIIPPHATLVFDVELLKLE 1fap B 2.7 BS01 RAP A 1 L2031 S2035 F2039 W2101 Y2105 F2108 L14 S18 F22 W84 Y88 F91 2.7.11.1 0044877 IC50=>10000nM, Kd=0.600000nM P42345 8662507 108 RVAILWHEMWHEGLEEASRLYFGERNVKGMFEVLEPLHAMMERGPQTLKETSFNQAYGRDLMEAQEWCRKYMKSGNVKDLTQAWDLYYHVFRRIS 1fkb A 1.7 BS01 RAP A 1 Y26 F36 D37 F46 Q53 E54 V55 I56 W59 Y82 F99 Y26 F36 D37 F46 Q53 E54 V55 I56 W59 Y82 F99 Y26 F36 D37 I56 Y82 F99 Y26 F36 D37 I56 Y82 F99 5.2.1.8 0000413,0003007,0003755,0005160,0005515,0005527,0005528,0005737,0005829,0006457,0006458,0014802,0014809,0016020,0016247,0016529,0022417,0030018,0030512,0030547,0032092,0032880,0032926,0033017,0034713,0042026,0042110,0043123,0044325,0050776,0055010,0060314,0060347,0070411,0070588,0070697,0097435,0098562,1902991,1990000,1990425 Kd=0.2nM -logKd/Ki=9.70, Kd=0.2nM IC50=0.600000nM, EC50=30nM, Ki=0.20nM P62942 108 GVQVETISPGDGRTFPKRGQTCVVHYTGMLEDGKKFDSSRDRNKPFKFMLGKQEVIRGWEEGVAQMSVGQRAKLTISPDYAYGATGHPGIIPPHATLVFDVELLKLE 1fkl A 1.7 BS01 RAP A 1 Y26 F36 D37 F46 Q53 E54 V55 W59 Y82 Y26 F36 D37 F46 Q53 E54 V55 W59 Y82 Y26 F36 D37 I56 Y82 F99 Y26 F36 D37 I56 Y82 F99 5.2.1.8 0000413,0001933,0003007,0003755,0005528,0005737,0005829,0006936,0007183,0016020,0016529,0019221,0019855,0030018,0031000,0031398,0032092,0032515,0032880,0032925,0033017,0042098,0042110,0042803,0043123,0044325,0046332,0048185,0050776,0051209,0051280,0055010,0060314,0060315,0060347,0070062,0097435,0098562,1902991,1990000,1990425 P18203 15299838 108 GVQVETISPGDGRTFPKRGQTCVVHYTGMLEDGKKFDSSRDRNKPFKFVLGKQEVIRGWEEGVAQMSVGQRAKLTISPDYAYGATGHPGIIPPNATLIFDVELLKLE 1pbk A 2.5 BS01 RAP A 1 Y135 D146 L162 G169 K170 V171 W175 Y198 I208 Y27 D38 L54 G61 K62 V63 W67 Y90 I100 Y135 F145 D146 I172 Y198 F216 Y27 F37 D38 I64 Y90 F108 5.2.1.8 0003755 Ki=0.9nM -logKd/Ki=9.05, Ki=0.9nM Q00688 225 PKYTKSVLKKGDKTNFPKKGDVVHCWYTGTLQDGTVFDTNIQTSAKKKKNAKPLSFKVGVGKVIRGWDEALLTMSKGEKARLEIEPEWAYGKKGQPDAKIPPNAKLTFEVELVDID 2dg3 A 1.7 BS01 RAP A 1 Y26 F36 D37 F46 Q53 E54 V55 I56 W59 Y82 H87 F99 Y26 F36 D37 F46 Q53 E54 V55 I56 W59 Y82 H87 F99 Y26 F36 D37 I56 Y82 F99 Y26 F36 D37 I56 Y82 F99 5.2.1.8 0000413,0003007,0003755,0005160,0005515,0005527,0005528,0005737,0005829,0006457,0006458,0014802,0014809,0016020,0016247,0016529,0022417,0030018,0030512,0030547,0032092,0032880,0032926,0033017,0034713,0042026,0042110,0043123,0044325,0050776,0055010,0060314,0060347,0070411,0070588,0070697,0097435,0098562,1902991,1990000,1990425 IC50=0.600000nM, EC50=30nM, Ki=0.20nM P62942 12600203 501 GVQVETISPGDGRTFPKRGQTCVVHYTGMLEDGKKFDSSRDRNKPFKFMLGKQEVIRGWEEGVAQMSVGQRAKLTISPDYAYGATGHPGIIPPHATLVFDVELLKLE 2dg4 A 1.7 BS01 RAP A 1 Y26 F36 D37 F46 Q53 E54 V55 F59 Y82 Y26 F36 D37 F46 Q53 E54 V55 F59 Y82 Y26 F36 D37 I56 Y82 F99 Y26 F36 D37 I56 Y82 F99 5.2.1.8 0000413,0003007,0003755,0005160,0005515,0005527,0005528,0005737,0005829,0006457,0006458,0014802,0014809,0016020,0016247,0016529,0022417,0030018,0030512,0030547,0032092,0032880,0032926,0033017,0034713,0042026,0042110,0043123,0044325,0050776,0055010,0060314,0060347,0070411,0070588,0070697,0097435,0098562,1902991,1990000,1990425 IC50=0.600000nM, EC50=30nM, Ki=0.20nM P62942 12600203 501 GVQVETISPGDGRTFPKRGQTCVVHYTGMLEDGKKFDSSRDRNKPFKFMLGKQEVIRGFEEGVAQMSVGQRAKLTISPDYAYGATGHPGIIPPHATLVFDVELLKLE 2dg9 A 1.7 BS01 RAP A 1 Y26 F36 D37 F46 Q53 E54 V55 I56 L59 Y82 H87 Y26 F36 D37 F46 Q53 E54 V55 I56 L59 Y82 H87 Y26 F36 D37 I56 Y82 F99 Y26 F36 D37 I56 Y82 F99 5.2.1.8 0000413,0003007,0003755,0005160,0005515,0005527,0005528,0005737,0005829,0006457,0006458,0014802,0014809,0016020,0016247,0016529,0022417,0030018,0030512,0030547,0032092,0032880,0032926,0033017,0034713,0042026,0042110,0043123,0044325,0050776,0055010,0060314,0060347,0070411,0070588,0070697,0097435,0098562,1902991,1990000,1990425 IC50=0.600000nM, EC50=30nM, Ki=0.20nM P62942 12600203 501 GVQVETISPGDGRTFPKRGQTCVVHYTGMLEDGKKFDSSRDRNKPFKFMLGKQEVIRGLEEGVAQMSVGQRAKLTISPDYAYGATGHPGIIPPHATLVFDVELLKLE 2vcd A -1.00 BS01 RAP A 1 Y55 F65 D66 F77 Q81 V82 I83 P84 W86 Y109 Y55 F65 D66 F77 Q81 V82 I83 P84 W86 Y109 Y55 F65 D66 I83 Y109 F126 Y55 F65 D66 I83 Y109 F126 5.2.1.8 0003755,0006457 Q5ZXE0 18366641 138 FNKKADENKVKGEAFLTENKNKPGVVVLPSGLQYKVINSGNGVKPGKSDTVTVEYTGRLIDGTVFDSTEKTGKPATFQVSQVIPGWTEALQLMPAGSTWEIYVPSGLAYGPRSVGGPIGPNETLIFKIHLISVKKSS 3kz7 A 1.95 BS01 RAP A 1 D146 L162 G169 K170 V171 I172 W175 Y198 D41 L57 G64 K65 V66 I67 W70 Y93 Y135 F145 D146 I172 Y198 F216 Y30 F40 D41 I67 Y93 F111 5.2.1.8 0003755 Q62446 24879919 225 EGPPKYTKSILKKGDKTNFPKKGDVVHCWYTGTLPDGTVFDTNIQTSSKKKKNAKPLSFKVGVGKVIRGWDEALLTMSKGEKARLEIEPEWAYGKKGQPDAKIPPNTKLIFEVELVDID 4drh A 2.3 BS01 RAP A 1 Y57 F67 D68 H71 F77 G84 Q85 V86 I87 W90 Y113 F130 Y49 F59 D60 H63 F69 G76 Q77 V78 I79 W82 Y105 F122 Y57 F67 D68 I87 Y113 F130 Y49 F59 D60 I79 Y105 F122 5.2.1.8 0003755 Ki=3.0nM Q13451 23358420 201 NNEESPTATVAEQGEDITSKKDRGVLKIVKRVGNGEETPMIGDKVYVHYKGKLSNGKKFDSSHDRNEPFVFSLGKGQVIKAWDIGVATMKKGEICHLLCKPEYAYGSAGSLPKIPSNATLFFEIELLDFKGE 4drh B 2.3 BS01 RAP A 1 S2035 F2039 T2098 W2101 Y2105 F2108 S18 F22 T81 W84 Y88 F91 2.7.11.1 0044877 IC50=>10000nM, Kd=0.600000nM P42345 23358420 201 AMDPEFMEMWHEGLEEASRLYFGERNVKGMFEVLEPLHAMMERGPQTLKETSFNQAYGRDLMEAQEWCRKYMKSGNVKDLTQAWDLYYHVFRRIS 4drh D 2.3 BS01 RAP D 1 Y57 F67 D68 H71 F77 G84 Q85 V86 I87 W90 Y113 F130 Y48 F58 D59 H62 F68 G75 Q76 V77 I78 W81 Y104 F121 5.2.1.8 0003755 Ki=3.0nM Q13451 23358420 201 NEESPTATVAEQGEDITSKKDRGVLKIVKRVGNGEETPMIGDKVYVHYKGKLSNGKKFDSSHDRNEPFVFSLGKGQVIKAWDIGVATMKKGEICHLLCKPEYAYGSAGSLPKIPSNATLFFEIELLDFKGE 4drh E 2.3 BS01 RAP D 1 L2031 S2035 R2036 F2039 W2101 Y2105 F2108 L13 S17 R18 F21 W78 Y82 F85 2.7.11.1 0044877 IC50=>10000nM, Kd=0.600000nM P42345 23358420 201 MDPEFMEMWHEGLEEASRLYFGERNVKGMFEVLEPLHAMMELKETSFNQAYGRDLMEAQEWCRKYMKSGNVKDLTQAWDLYYHVFRRIS 4dri A 1.45 BS01 RAP A 1 Y57 D68 R73 F77 G84 Q85 V86 I87 W90 Y113 Y38 D49 R54 F58 G65 Q66 V67 I68 W71 Y94 Y57 F67 D68 I87 Y113 F130 Y38 F48 D49 I68 Y94 F111 5.2.1.8 0003755 Ki=3.0nM Q13451 23358420 201 EQGEDITSKKDRGVLKIVKRVGNGEETPMIGDKVYVHYKGKLSNGKKFDSSHDRNEPFVFSLGKGQVIKAWDIGVATMKKGEICHLLCKPEYAYGSAGSLPKIPSNATLFFEIELLDFKGE 4dri B 1.45 BS01 RAP A 1 L2031 S2035 F2039 T2098 Y2105 F2108 L15 S19 F23 T82 Y89 F92 2.7.11.1 0044877 IC50=>10000nM, Kd=0.600000nM P42345 23358420 201 GAMDPEFMEMWHEGLEEASRLYFGERNVKGMFEVLEPLHAMMERGPQTLKETSFNQAYGRDLMEAQEWCRKYMKSGNVKDLTQAWDLYYHVFRRIS 4drj A 1.8 BS01 RAP A 1 Y57 D68 F77 G84 E85 V86 I87 W90 Y113 K121 Y39 D50 F59 G66 E67 V68 I69 W72 Y95 K103 Y57 F67 D68 I87 Y113 F130 Y39 F49 D50 I69 Y95 F112 5.2.1.8 0003755 Q02790 23358420 201 PMEGVDISPKQDEGVLKVIKREGTGTEMPMIGDRVFVHYTGWLLDGTKFDSSLDRKDKFSFDLGKGEVIKAWDIAIATMKVGEVCHITCKPEYAYGSAGSPPKIPPNATLVFEVELFEFKG 4drj B 1.8 BS01 RAP A 1 L2031 S2035 F2039 T2098 Y2105 F2108 L13 S17 F21 T80 Y87 F90 2.7.11.1 0044877 IC50=>10000nM, Kd=0.600000nM P42345 23358420 201 MDPEFMEMWHEGLEEASRLYFGERNVKGMFEVLEPLHAMMERGPQTLKETSFNQAYGRDLMEAQEWCRKYMKSGNVKDLTQAWDLYYHVFRRISKQ 4qt2 A 1.44 BS01 RAP A 1 Y44 D56 F65 G72 E73 V74 I75 W78 Y101 Y38 D50 F59 G66 E67 V68 I69 W72 Y95 Y44 F55 D56 I75 Y101 F118 Y38 F49 D50 I69 Y95 F112 5.2.1.8 0003755 ic50=0.48uM -logKd/Ki=6.32, IC50=0.48uM Q8I4V8 26057671 202 FEKVELTADGGVIKTILKKGDEGEENIPKKGNEVTVHYVGKLESTGKVFDSSFDRNVPFKFHLEQGEVIKGWDICVSSMRKNEKCLVRIESMYGYGDEGCGESIPGNSVLLFEIELLSFREL 4qt3 A 1.4 BS01 RAP A 1 Y44 F55 D56 F65 E73 V74 I75 W78 Y101 F118 Y40 F51 D52 F61 E69 V70 I71 W74 Y97 F114 Y44 F55 D56 I75 Y101 F118 Y40 F51 D52 I71 Y97 F114 5.2.1.8 0003755 ic50=0.48uM Q8I4V8 26057671 202 QEFEKVELTADGGVIKTILKKGDEGEENIPKKGNEVTVHYVGKLESTGKVFDSSFDRNVPFKFHLEQGEVIKGWDICVSSMRKNEKCLVRIESMYGYGDEGCGESIPGNSVLLFEIELLSFRELE 5flc B 5.9 BS01 RAP C 1 E2032 S2035 R2036 F2039 G2040 W2101 Y2105 F2108 E588 S591 R592 F595 G596 W657 Y661 F664 2.7.11.1 0004674,0016301,0044877 IC50=>10000nM, Kd=0.600000nM P42345 26678875 999 YAKALHYKELEFQKGPTPAILESLISINNKLQQPEAAAGVLEYAMKHFGELEIQATWYEKLHEWEDALVAYDKKMDTNKDDPELMLGRMRCLEALGEWGQLHQQCCEKWTLVNDETQAKMARMAAAAAWGLGQWDSMEEYTCMIPRDTHDGAFYRAVLALHQDLFSLAQQCIDKARDLLDAELTAMAGESYSRAYGAMVSCHMLSELEEVIQYKLVPERREIIRQIWWERLQGCQRIVEDWQKILMVRSLVVSPHEDMRTWLKYASLCGKSGRLALAHKTLVLLLGVDPSRQLDHPLPTVHPQVTYAYMKNMWKSARKIDAFQHMQHFVQTMQQQAQHAIATEDQQHKQELHKLMARCFLKLGEWQLNLQGINESTIPKVLQYYSAATEHDRSWYKAWHAWAVMNFEAVLHYKHQNQARDEKKKVTEDLSKTLLMYTVPAVQGFFRSISLSRGNNLQDTLRVLTLWFDYGHWPDVNEALVEGVKAIQIDTWLQVIPQLIARIDTPRPLVGRLIHQLLTDIGRYHPQALIYPLTVASKSTTTARHNAANKILKNMCEHSNTLVQQAMMVSEELIRVAILWHEMWHEGLEEASRLYFGERNVKGMFEVLEPLHAMMERGPQTLKETSFNQAYGRDLMEAQEWCRKYMKSGNVKDLTQAWDLYYHVFRRISKQLPQLTSLELQYVSPKLLMCRDLELAVPGTYDPNQPIIRIQSIAPSLQVITSKQRPRKLTLMGSNGHEFVFLLKGHEDLRQDERVMQLFGLVNTLLANDPTSLRKNLSIQRYAVIPLSTNSGLIGWVPHCDTLHALIRDYREKKKILLNIEHRIMLRMAPDYDHLTLMQKVEVFEHAVNNTAGDDLAKLLWLKSPSSEVWFDRRTNYTRSLAVMSMVGYILGLGDRHPSNLMLDRLSGKILHIDFGDCFEVAMTREKFPEKIPFRLTRMLTNAMEVTGLDGNYRITCHTVMEVLREHKDSVMAVLEAFVYDPLLNWRLMDTNTALNKKAIQIINRVRDKLTGRDFSHDDTLDVPTQVELLIKQATSHENLCQCYIGWCPFW 5flc C 5.9 BS01 RAP C 1 X54 X55 X56 X54 X55 X56 26678875 999 PPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPP 5flc F 5.9 BS01 RAP G 1 E2032 S2035 R2036 F2039 G2040 W2101 Y2105 F2108 E588 S591 R592 F595 G596 W657 Y661 F664 2.7.11.1 0004674,0016301,0044877 IC50=>10000nM, Kd=0.600000nM P42345 26678875 999 YAKALHYKELEFQKGPTPAILESLISINNKLQQPEAAAGVLEYAMKHFGELEIQATWYEKLHEWEDALVAYDKKMDTNKDDPELMLGRMRCLEALGEWGQLHQQCCEKWTLVNDETQAKMARMAAAAAWGLGQWDSMEEYTCMIPRDTHDGAFYRAVLALHQDLFSLAQQCIDKARDLLDAELTAMAGESYSRAYGAMVSCHMLSELEEVIQYKLVPERREIIRQIWWERLQGCQRIVEDWQKILMVRSLVVSPHEDMRTWLKYASLCGKSGRLALAHKTLVLLLGVDPSRQLDHPLPTVHPQVTYAYMKNMWKSARKIDAFQHMQHFVQTMQQQAQHAIATEDQQHKQELHKLMARCFLKLGEWQLNLQGINESTIPKVLQYYSAATEHDRSWYKAWHAWAVMNFEAVLHYKHQNQARDEKKKVTEDLSKTLLMYTVPAVQGFFRSISLSRGNNLQDTLRVLTLWFDYGHWPDVNEALVEGVKAIQIDTWLQVIPQLIARIDTPRPLVGRLIHQLLTDIGRYHPQALIYPLTVASKSTTTARHNAANKILKNMCEHSNTLVQQAMMVSEELIRVAILWHEMWHEGLEEASRLYFGERNVKGMFEVLEPLHAMMERGPQTLKETSFNQAYGRDLMEAQEWCRKYMKSGNVKDLTQAWDLYYHVFRRISKQLPQLTSLELQYVSPKLLMCRDLELAVPGTYDPNQPIIRIQSIAPSLQVITSKQRPRKLTLMGSNGHEFVFLLKGHEDLRQDERVMQLFGLVNTLLANDPTSLRKNLSIQRYAVIPLSTNSGLIGWVPHCDTLHALIRDYREKKKILLNIEHRIMLRMAPDYDHLTLMQKVEVFEHAVNNTAGDDLAKLLWLKSPSSEVWFDRRTNYTRSLAVMSMVGYILGLGDRHPSNLMLDRLSGKILHIDFGDCFEVAMTREKFPEKIPFRLTRMLTNAMEVTGLDGNYRITCHTVMEVLREHKDSVMAVLEAFVYDPLLNWRLMDTNTALNKKAIQIINRVRDKLTGRDFSHDDTLDVPTQVELLIKQATSHENLCQCYIGWCPFW 5flc G 5.9 BS01 RAP G 1 X54 X55 X56 X54 X55 X56 26678875 999 PPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPPP 5gpg A 1.67 BS01 RAP A 1 Y135 D146 L162 G169 K170 V171 W175 Y198 F216 Y28 D39 L48 G55 K56 V57 W61 Y84 F102 Y135 F145 D146 I172 Y198 F216 Y28 F38 D39 I58 Y84 F102 5.2.1.8 0003755 Q00688 27610411 301 SPKYTKSVLKKGDKTNFPKKGDVVHCWYTGTLQDGTVFDTNIQNAKPLSFKVGVGKVIRGWDEALLTMSKGEKARLEIEPEWAYGKKGQPDAKIPPNAKLTFEVELVDID 5gpg B 1.67 BS01 RAP A 1 L2031 S2035 R2036 F2039 T2098 D2102 Y2105 F2108 L12 S16 R17 F20 T79 D83 Y86 F89 2.7.11.1 0044877 IC50=>10000nM, Kd=0.600000nM P42345 27610411 301 SILWHEMWHEGLEEASRLYFGERNVKGMFEVLEPLHAMMERGPQTLKETSFNQAYGRDLMEAQEWCRKYMKSGNVKDLTQAWDLYYHVFRRIS 5hkg A 1.5 BS01 RAP A 1 Y26 F36 D37 F46 Q53 E54 V55 I56 F59 Y82 Y26 F36 D37 F46 Q53 E54 V55 I56 F59 Y82 Y26 F36 D37 I56 Y82 F99 Y26 F36 D37 I56 Y82 F99 5.2.1.8 0002027,0003755,0005102,0005219,0005515,0005528,0005737,0006458,0006939,0007204,0009749,0010459,0010880,0010881,0016020,0016247,0016529,0019227,0019722,0019855,0022417,0030018,0030073,0030551,0033017,0033197,0034704,0035773,0042026,0042098,0042542,0044325,0048680,0050849,0051209,0051280,0051284,0051775,0060314,0061179 Kd=0.200000nM P68106 27670942 201 GVEIETISPGDGRTFPKKGQTCVVHYTGMLQNGKKFDSSRDRNKPFKFRIGKQEVIKGFEEGAAQMSLGQRAKLTCTPDVAYGATGHPGVIPPNATLIFDVELLNLE 6m4u A 2.2 BS01 RAP A 1 Y27 F37 D38 F47 Q54 E55 V56 I57 W60 Y83 I92 Y27 F37 D38 F47 Q54 E55 V56 I57 W60 Y83 I92 5.2.1.8 0000413,0003007,0003755,0005160,0005515,0005527,0005528,0005737,0005829,0006457,0006458,0014802,0014809,0016020,0016247,0016529,0022417,0030018,0030512,0030547,0032092,0032880,0032926,0033017,0034713,0042026,0042110,0043123,0044325,0050776,0055010,0060314,0060347,0070411,0070588,0070697,0097435,0098562,1902991,1990000,1990425 IC50=0.600000nM, EC50=30nM, Ki=0.20nM P62942 32747768 201 MGVQVETISPGDGRTFPKRGQTCVVHYTGMLEDGKKFDSSRDRNKPFKFMLGKQEVIRGWEEGVAQMSVGQRAKLTISPDYAYGATGHPGIIPPHATLVFDVELLKLE 6m4u B 2.2 BS01 RAP A 1 L2031 E2032 S2035 F2039 Y2105 F2108 L11 E12 S15 F19 Y85 F88 2.7.11.1 0044877 IC50=>10000nM, Kd=0.600000nM P42345 32747768 201 ILWHEMWHEGLEEASRLYFGERNVKGMFEVLEPLHAMMERGPQTLKETSFNQAYGRDLMEAQEWCRKYMKSGNVKDLLQAWDLYYHVFRRISK 6m4u E 2.2 BS01 RAP E 1 Y27 F37 D38 F47 E55 V56 I57 W60 Y83 I92 Y29 F39 D40 F49 E57 V58 I59 W62 Y85 I94 5.2.1.8 0000413,0003007,0003755,0005160,0005515,0005527,0005528,0005737,0005829,0006457,0006458,0014802,0014809,0016020,0016247,0016529,0022417,0030018,0030512,0030547,0032092,0032880,0032926,0033017,0034713,0042026,0042110,0043123,0044325,0050776,0055010,0060314,0060347,0070411,0070588,0070697,0097435,0098562,1902991,1990000,1990425 IC50=0.600000nM, EC50=30nM, Ki=0.20nM P62942 32747768 201 GSMGVQVETISPGDGRTFPKRGQTCVVHYTGMLEDGKKFDSSRDRNKPFKFMLGKQEVIRGWEEGVAQMSVGQRAKLTISPDYAYGATGHPGIIPPHATLVFDVELLKLE 6m4u F 2.2 BS01 RAP E 1 L2031 E2032 S2035 F2039 L2098 D2102 Y2105 F2108 L13 E14 S17 F21 L80 D84 Y87 F90 2.7.11.1 0044877 IC50=>10000nM, Kd=0.600000nM P42345 32747768 201 GSILWHEMWHEGLEEASRLYFGERNVKGMFEVLEPLHAMMERGPQTLKETSFNQAYGRDLMEAQEWCRKYMKSGNVKDLLQAWDLYYHVFRRISK 6m4v B 2.92 BS01 RAP B 1 F37 D38 F47 Q54 E55 V56 I57 W60 Y83 I91 F100 F4 D5 F14 Q21 E22 V23 I24 W27 Y50 I58 F67 5.2.1.8 0003755 IC50=0.600000nM, EC50=30nM, Ki=0.20nM P62942 32747768 201 GKKFDSSRDRNKPFKFMLGKQEVIRGWEEGVAQMSVGQRAKLTISPDYAYGATGHPGIIPPHATLVFDVELLKLE 6m4v D 2.92 BS01 RAP D 1 F37 D38 F47 Q54 E55 V56 I57 W60 Y83 I91 F100 F4 D5 F14 Q21 E22 V23 I24 W27 Y50 I58 F67 5.2.1.8 0003755 IC50=0.600000nM, EC50=30nM, Ki=0.20nM P62942 32747768 201 GKKFDSSRDRNKPFKFMLGKQEVIRGWEEGVAQMSVGQRAKLTISPDYAYGATGHPGIIPPHATLVFDVELLKLE 6m4w A 3.11 BS03 RAP F 1 A-197 K-195 A174 K176 5.2.1.8 0003755,0005515,0006974,0008643,0015144,0015768,0016020,0030288,0034219,0034289,0042597,0042956,0043190,0055052,0055085,0060326,1901982,1990060 P0AEX9,P62942 32747768 201 MKIEEGKLVIWINGDKGYNGLAEVGKKFEKDTGIKVTVEHPDKLEEKFPQVAATGDGPDIIFWAHDRFGGYAQSGLLAEITPAAAFQDKLYPFTWDAVRYNGKLIAYPIAVEALSLIYNKDLLPNPPKTWEEIPALDKELKAKGKSALMFNLQEPYFTWPLIAADGGYAFKYAAGKYDIKDVGVDNAGAKAGLTFLVDLIKNKHMNADTDYSIAEAAFNKGETAMTINGPWAWSNIDTSAVNYGVTVLPTFKGQPSKPFVGVLSAGINAASPNKELAKEFLENYLLTDEGLEAVNKDKPLGAVALKSYEEELAKDPRIAATMENAQKGEIMPNIPQMSAFWYAVRTAVINAASGRQTVDEALKDAQTNAAAMGVQVETISPGDGRTFPKRGQTCVVHYTGMLE 6m4w D 3.11 BS01 RAP D 1 D38 F47 E55 V56 W60 Y83 I91 D5 F14 E22 V23 W27 Y50 I58 5.2.1.8 0003755 IC50=0.600000nM, EC50=30nM, Ki=0.20nM P62942 32747768 201 GKKFDSSRDRNKPFKFMLGKQEVIRGWEEGVAQMSVGQRAKLTISPDYAYGATGHPGIIPPHATLVFDVELLKLE 6m4w E 3.11 BS01 RAP E 1 F37 D38 F47 E55 V56 I57 W60 Y83 F5 D6 F15 E23 V24 I25 W28 Y51 5.2.1.8 0003755 IC50=0.600000nM, EC50=30nM, Ki=0.20nM P62942 32747768 201 DGKKFDSSRDRNKPFKFMLGKQEVIRGWEEGVAQMSVGQRAKLTISPDYAYGATGHPGIIPPHATLVFDVELLKLE 6m4w F 3.11 BS01 RAP F 1 F37 D38 E55 V56 W60 Y83 I91 F5 D6 E23 V24 W28 Y51 I59 5.2.1.8 0003755 IC50=0.600000nM, EC50=30nM, Ki=0.20nM P62942 32747768 201 DGKKFDSSRDRNKPFKFMLGKQEVIRGWEEGVAQMSVGQRAKLTISPDYAYGATGHPGIIPPHATLVFDVELLKLE 6m4w G 3.11 BS01 RAP D 1 L2031 S2035 R2036 F2039 L2098 W2101 Y2105 F2108 L12 S16 R17 F20 L79 W82 Y86 F89 2.7.11.1 0044877 IC50=>10000nM, Kd=0.600000nM P42345 32747768 201 SILWHEMWHEGLEEASRLYFGERNVKGMFEVLEPLHAMMERGPQTLKETSFNQAYGRDLMEAQEWCRKYMKSGNVKDLLQAWDLYYHVFRRIS 6m4w H 3.11 BS01 RAP E 1 L2031 S2035 F2039 L2098 Y2105 F2108 L12 S16 F20 L79 Y86 F89 2.7.11.1 0044877 IC50=>10000nM, Kd=0.600000nM P42345 32747768 201 SILWHEMWHEGLEEASRLYFGERNVKGMFEVLEPLHAMMERGPQTLKETSFNQAYGRDLMEAQEWCRKYMKSGNVKDLLQAWDLYYHVFRRIS 6m4w I 3.11 BS01 RAP F 1 L2031 S2035 R2036 F2039 L2098 W2101 Y2105 F2108 L12 S16 R17 F20 L79 W82 Y86 F89 2.7.11.1 0044877 IC50=>10000nM, Kd=0.600000nM P42345 32747768 201 SILWHEMWHEGLEEASRLYFGERNVKGMFEVLEPLHAMMERGPQTLKETSFNQAYGRDLMEAQEWCRKYMKSGNVKDLLQAWDLYYHVFRRIS 7f2j A 1.6 BS01 RAP A 1 D408 F416 G423 S424 V425 I426 W429 Y452 D47 F55 G62 S63 V64 I65 W68 Y91 5.2.1.8 0003755 Q93ZG9 35218805 501 SQVRTYPNGLIVEELSMGKPNGKRADPGKTVSVRYIGKLQKNGKIFDSNIGKSPFKFRLGIGSVIKGWDVGVNGMRVGDKRKLTIPPSMGYGVKGAGGQIPPNSWLTFDVELINVQL 7f2j B 1.6 BS01 RAP B 1 Y396 F407 D408 F416 G423 S424 V425 I426 W429 Y452 Y34 F45 D46 F54 G61 S62 V63 I64 W67 Y90 5.2.1.8 0003755 Q93ZG9 35218805 501 QVRTYPNGLIVEELSMGKPNGKRADPGKTVSVRYIGKLQKNGKIFDSNIGKSPFKFRLGIGSVIKGWDVGVNGMRVGDKRKLTIPPSMGYGVKGAGGQIPPNSWLTFDVELINVQL 8xi9 A 1.85 BS01 RAP A 1 Y121 D132 F141 Q148 E149 V150 I151 W154 Y177 Y120 D131 F140 Q147 E148 V149 I150 W153 Y176 P42345,P62942 39031920 301 GWHEMWHEGLEEASRLYFGERNVKGMFEVLEPLHAMMERGPQTLKETSFNQAYGRDLMEAQEWCRKYMKSGNVKDLTQAWDLYYHVFRRISKQMGVQVETISPGDGRTFPKRGQTCVVHYTGMLEDGKKFDSSRDRNKPFKFMLGKQEVIRGWEEGVAQMSVGQRAKLTISPDYAYGATGHPGIIPPHATLVFDVELLKLE