4rqv A 1.502 BS02 R2S A 1 K115 I118 I119 V124 T128 R131 T148 L155 F157 K45 I48 I49 V54 T58 R61 T78 L85 F87 D205 K207 E209 N210 D223 T245 D135 K137 E139 N140 D153 T175 2.7.11.1 0004672,0004674,0005524,0006468 -logKd/Ki=5.05, Kd=9uM O15530 25518860 406 PPQPRKKRPEDFKFGKILGEGSFSTVVLARELATSREYAIKILEKRHIIKENKVPYVTRERDVMSRLDHPFFVKLYFTFQDDEKLYFGLSYAKNGELLKYIRKIGSFDETCTRFYTAEIVSALEYLHGKGIIHRDLKPENILLNEDMHIQITDFGTAKVLSPESKQARANSFVGTAQYVSPELLTEKSACKSSDLWALGCIIYQLVAGLPPFRAGNEGLIFAKIIKLEYDFPEKFFPKARDLVEKLLVLDATKRLGCEEMEGYGPLKAHPFFESVTWENLHQQTPPKLT