4mpn A 1.752 BS01 PV0 A 1 N255 R258 A259 E262 D290 G294 V295 T354 N240 R243 A244 E247 D275 G279 V280 T323 H247 E251 K254 N255 H232 E236 K239 N240 2.7.11.2 0004672,0004740,0005515,0005524,0005654,0005739,0005759,0005829,0006006,0006111,0006885,0008286,0010510,0010565,0010906,0016301,0016310,0031670,0034614,0042593,0042803,0045254,0050848,0072332 Kd=239nM -logKd/Ki=6.62, Kd=239nM EC50=456nM, Kd=156nM, IC50=456nM Q15119 24356970 501 SLAGAPKYIEHFSKFSPSPLSMKQFLDFGSSNACEKTSFTFLRQELPVRLANIMKEINLLPDRVLSTPSVQLVQSWYVQSLLDIMEFLDKDPEDHRTLSQFTDALVTIRNRHNDVVPTMAQGVLEYKDTYGDDPVSNQNIQYFLDRFYLSRISIRMLINQHTLIFDPAHPKHIGSIDPNCNVSEVVKDAYDMAKLLCDKYYMASPDLEIQEINAANSKQPIHMVYVPSHLYHMLFELFKNAMRATVESHESSLILPPIKVMVALGEEDLSIKMSDRGGGVPLRKIERLFSYMYSTGYGLPISRLYAKYFQGDLQLFSMEGFGTDAVIYLKALSTDSVERLPVYNKSAWRHYQTIQEAGDWCVP