2zk1 A 2.61 BS01 PTG A 1 C285 R288 S289 Y327 L330 L333 L340 M364 K367 H449 L453 Y473 C83 R86 S87 Y125 L128 L131 L138 M162 K165 H247 L251 Y271 ? 0003677,0004879,0005634,0006355 P37231 18977231 1 QLNPESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHITPLQEQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL 2zk1 B 2.61 BS01 PTG B 1 C285 R288 H323 I326 L330 L333 K367 H449 C79 R82 H117 I120 L124 L127 K161 H243 ? 0003677,0004879,0005634,0006355 P37231 18977231 2 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHITPLQEQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETHPLLQEIY 2zk2 A 2.26 BS02 PTG A 1 C285 S289 H323 I326 M329 L330 M364 H449 L469 Y473 C83 S87 H121 I124 M127 L128 M162 H247 L267 Y271 ? 0003677,0004879,0005634,0006355 P37231 18977231 477 QLNPESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHITPLQEQSKEVAIRIFQGCQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL 2zvt A 1.9 BS01 PTG A 1 R288 S289 H323 I326 Y327 I341 M364 H449 L469 Y473 R86 S87 H121 I124 Y125 I139 M162 H247 L267 Y271 ? 0003677,0004879,0005634,0006355 P37231 19101554 1 QLNPESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHITPLQEQSKEVAIRIFQGSQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETDMSLHPLLQEIYKDL 2zvt B 1.9 BS01 PTG B 1 S285 R288 A292 L330 I341 S342 E343 M348 F363 M364 S79 R82 A86 L124 I135 S136 E137 M142 F157 M158 ? 0003677,0004879,0005634,0006355 P37231 19101554 2 ESADLRALAKHLYDSYIKSFPLTKAKARAILTGKTTDKSPFVIYDMNSLMMGEDKIKFKHITPLQEQSKEVAIRIFQGSQFRSVEAVQEITEYAKSIPGFVNLDLNDQVTLLKYGVHEIIYTMLASLMNKDGVLISEGQGFMTREFLKSLRKPFGDFMEPKFEFAVKFNALELDDSDLAIFIAVIILSGDRPGLLNVKPIEDIQDNLLQALELQLKLNHPESSQLFAKLLQKMTDLRQIVTEHVQLLQVIKKTETHPLLQEIY 6i5g A 2.0 BS01 PTG A 1 F387 S415 L417 M419 D496 F497 V498 H524 W525 F158 S186 L188 M190 D267 F268 V269 H295 W296 F267 D335 W336 D496 H524 F38 D106 W107 D267 H295 3.1.3.76,3.3.2.10 0003824 Ki=8.56uM -logKd/Ki=4.89, Ki=13.03uM P34913 31123712 607 TSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSD 6i5g B 2.0 BS01 PTG B 1 Y383 F387 M419 D496 F497 V498 H524 Y154 F158 M190 D267 F268 V269 H295 F267 D335 W336 D496 H524 F38 D106 W107 D267 H295 3.1.3.76,3.3.2.10 0003824 Ki=8.56uM P34913 31123712 607 TSCNPSDMSHGYVTVKPRVRLHFVELGSGPAVCLCHGFPESWYSWRYQIPALAQAGYRVLAMDMKGYGESSAPPEIEEYCMEVLCKEMVTFLDKLGLSQAVFIGHDWGGMLVWYMALFYPERVRAVASLNTPFIPANPNMSPLESIKANPVFDYQLYFQEPGVAEAELEQNLSRTFKSLFRASDESVLSMHKVCEAGGLFVNSPEEPSLSRMVTEEEIQFYVQQFKKSGFRGPLNWYRNMERNWKWACKSLGRKILIPALMVTAEKDFVLVPQMSQHMEDWIPHLKRGHIEDCGHWTQMDKPTEVNQILIKWLDSD