3el8 A 2.3 BS01 PD5 A 1 V281 A293 E310 M314 Y340 M341 L393 A403 D404 V24 A36 E53 M57 Y83 M84 L136 A146 D147 D386 R388 A390 N391 D404 F424 D129 R131 A133 N134 D147 F154 2.7.10.2 0004672,0004713,0005524,0006468 ic50=25nM -logKd/Ki=7.60, IC50=25nM P00523 18940662 601 DAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLKPGTMSPEAFLQEAQVMKKLRHEKLVQLYAVVSEEPIYIVTEYMSKGSLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFGLARLFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 3qlf A 2.75 BS01 PD5 A 1 V281 A293 M314 Y340 M341 L393 A403 D404 F405 V24 A36 M48 Y74 M75 L127 A137 D138 F139 D386 R388 A390 N391 D404 F424 D120 R122 A124 N125 D138 F140 2.7.10.2 0004672,0004713,0005524,0006468 P00523 601 DAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLKLQEAQVMKKIRHEKLVQLYAVVSEEPIYIVTEYMSKGSLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL 3qlf B 2.75 BS01 PD5 B 1 A293 K295 L297 E310 M314 I336 Y340 M341 L393 A36 K38 L40 E51 M55 I77 Y81 M82 L134 D386 R388 A390 N391 D404 F424 D127 R129 A131 N132 D145 F149 2.7.10.2 0004672,0004713,0005524,0006468 P00523 601 DAWEIPRESLRLEVKLGQGCFGEVWMGTWNGTTRVAIKTLKPMSPEAFLQEAQVMKKIRHEKLVQLYAVVSEEPIYIVTEYMSKGSLLDFLKGEMGKYLRLPQLVDMAAQIASGMAYVERMNYVHRDLRAANILVGENLVCKVADFARFPIKWTAPEAALYGRFTIKSDVWSFGILLTELTTKGRVPYPGMVNREVLDQVERGYRMPCPPECPESLHDLMCQCWRKDPEERPTFEYLQAFLEDYFTSTEPQYQPGENL