2qoh A 1.95 BS01 P3Y A 1 G249 Y253 V256 A269 V299 T315 M318 G321 N322 L370 G22 Y26 V29 A42 V69 T85 M88 G91 N92 L140 D363 A365 R367 N368 D381 P402 D133 A135 R137 N138 D151 P172 2.7.10.2 0004672,0004713,0005524,0006468 -logKd/Ki=7.70, IC50=20nM P00520 17718712 1 GSPNYDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKEEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVSAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQESS 2qoh B 1.95 BS01 P3Y B 1 L248 G249 Y253 V256 A269 T315 M318 G321 N322 L370 D381 L21 G22 Y26 V29 A42 T85 M88 G91 N92 L140 D151 D363 A365 R367 N368 D381 P402 D133 A135 R137 N138 D151 P172 2.7.10.2 0004672,0004713,0005524,0006468 P00520 17718712 1 GSPNYDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKMEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIITEFMTYGNLLDYLRECNRQEVSAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQESSISDEVEKELG 2z60 A 1.95 BS01 P3Y A 1 L248 G249 Y253 V256 A269 F317 M318 G321 N322 L370 L21 G22 Y26 V29 A42 F87 M88 G91 N92 L140 D363 A365 R367 N368 D381 P402 D133 A135 R137 N138 D151 P172 2.7.10.2 0004672,0004713,0005524,0006468 -logKd/Ki=8.05, IC50=9nM P00520 17718712 1 GSPNYDKWEMERTDITMKHKLGGGQYGEVYEGVWKKYSLTVAVKTLKEEVEEFLKEAAVMKEIKHPNLVQLLGVCTREPPFYIIIEFMTYGNLLDYLRECNRQEVSAVVLLYMATQISSAMEYLEKKNFIHRDLAARNCLVGENHLVKVADFGLSRLMTGDTYTAHAGAKFPIKWTAPESLAYNKFSIKSDVWAFGVLLWEIATYGMSPYPGIDLSQVYELLEKDYRMERPEGCPEKVYELMRACWQWNPSDRPSFAEIHQAFETMFQESSISDEVEKELG