1ikt A 1.75 BS01 OXN A 1 W36 F79 Q90 F93 S107 Q108 Q111 W31 F74 Q85 F88 S102 Q103 Q106 1.1.1.n12,4.2.1.107,4.2.1.119 -logKd/Ki=3.40, Kd=400uM P51659 11700068 123 LQSTFVFEEIGRRLKDIGPEVVKKVNAVFEWHITKGGNIGAKWTIDLKSGSGKVYQGPAKGAADTTIILSDEDFMEVVLGKLDPQKAFFSGRLKARGNIMLSQKLQMILKDYAKL 1ueh B 1.73 BS03 OXN B 1 V50 R51 V54 S55 E96 L100 H103 V34 R35 V38 S39 E80 L84 H87 D26 H43 L137 D10 H27 L121 2.5.1.31 0000287,0005737,0005829,0008360,0008834,0009252,0016094,0016740,0016765,0036094,0042803,0043164,0045547,0046872,0051301,0071555 P60472 12756244 801 GCRHVAIIMDGNGRWAKKQGKIRAFGHKAGAKSVRRAVSFAANNGIEALTLYAFSSENWNRPAQEVSALMELFVWALDSEVKSLHRHNVRLRIIGDTSRFNSRLQERIRKSEALTAGNTGLTLNIAANYGGRWDIVQGVRQLAEKVQQGNLQPDQIDEEMLNQHVCMHELAPVDLVIRTGGEHRISNFLLWQIAYAELYFTDVLWPDFDEQDFEGALNAFANRER 1ueh B 1.73 BS04 OXN B 2 M25 N28 G46 A69 W221 M9 N12 G30 A53 W205 D26 H43 L137 D10 H27 L121 2.5.1.31 0000287,0005737,0005829,0008360,0008834,0009252,0016094,0016740,0016765,0036094,0042803,0043164,0045547,0046872,0051301,0071555 P60472 12756244 802 GCRHVAIIMDGNGRWAKKQGKIRAFGHKAGAKSVRRAVSFAANNGIEALTLYAFSSENWNRPAQEVSALMELFVWALDSEVKSLHRHNVRLRIIGDTSRFNSRLQERIRKSEALTAGNTGLTLNIAANYGGRWDIVQGVRQLAEKVQQGNLQPDQIDEEMLNQHVCMHELAPVDLVIRTGGEHRISNFLLWQIAYAELYFTDVLWPDFDEQDFEGALNAFANRER 2d4q A 2.3 BS01 OXN A 1 F1633 W1641 F74 W82 ? P21359 16397625 701 KEEFKALKTLSIFYQAGTSKAGNPIFYYVARRFKTGQINGDLLIYHVLLTLKPYYAKPYEIVVDLTHTGPSNRFKTDFLSKWFVVFPGFAYDNVSAVYIYNCNSWVREYTKYHERLLTGLKGSKRLVFIDCPGKLAEHIEHEQQKLPAATLALEEDLKVFHNALKLAHKDTKVSIKVGSTAVQVTSAERTKVLGQSVFLNDIYYASEIEEICLVDENQFTLTIANQGTPLTFMHQECEAIVQSIIHIRTRWELSQPD 2d4q B 2.3 BS01 OXN B 1 Y1587 V1622 F1633 W1641 Y1668 Y28 V63 F74 W82 Y109 ? P21359 16397625 702 KEEFKALKTLSIFYQAGTSKAGNPIFYYVARRFKTGQINGDLLIYHVLLTLKPYYAKPYEIVVDLTHTGPSNRFKTDFLSKWFVVFPGFAYDNVSAVYIYNCNSWVREYTKYHERLLTGLSKRLVFIDCPGKLAEHIEHEQQKLPAATLALEEDLKVFHNALKLAHKDTKVSIKVGSTAVQVTSAERTKVLGQSVFLNDIYYASEIEEICLVDENQFTLTIANQGTPLTFMHQECEAIVQSIIHIRTRWELSQPD 2q32 A 2.4 BS01 OXN A 1 A48 E49 V54 F57 L74 Y134 T155 R156 L167 Y187 F227 N230 F234 A20 E21 V26 F29 L46 Y106 T127 R128 L139 Y159 F199 N202 F206 N50 Y78 T155 R156 G159 D160 G164 N22 Y50 T127 R128 G131 D132 G136 1.14.14.18 0004392,0006788 P30519 17965015 301 RMADLSELLKEGTKEAHDRAENTQFVKDFLKGNIKKELFKLATTALYFTYSALEEEMERNKDHPAFAPLYFPMELHRKEALTKDMEYFFGENWEEQVQAPKAAQKYVERIHYIGQNEPELLVAHAYTRYMGDLSGGQVLKKVAQRALKLPSTGEGTQFYLFENVDNAQQFKQLYRARMNALDLNMKTKERIVEEANKAFEYNMQIFNELDQAG 2q32 B 2.4 BS01 OXN B 1 V54 L74 Y134 R156 G159 D160 G163 L167 A226 F227 N230 I233 F234 V24 L44 Y104 R126 G129 D130 G133 L137 A196 F197 N200 I203 F204 N50 Y78 T155 R156 G159 D160 G164 N20 Y48 T125 R126 G129 D130 G134 1.14.14.18 0004392,0006788 P30519 17965015 301 ADLSELLKEGTKEAHDRAENTQFVKDFLKGNIKKELFKLATTALYFTYSALEEEMERNKDHPAFAPLYFPMELHRKEALTKDMEYFFGENWEEQVQAPKAAQKYVERIHYIGQNEPELLVAHAYTRYMGDLSGGQVLKKVAQRALKLPSTGEGTQFYLFENVDNAQQFKQLYRARMNALDLNMKTKERIVEEANKAFEYNMQIFNELDQAGSTLARET 4tpl A 2.9 BS01 OXN A 1 T2 C15 T13 C26 3.4.21.91,3.6.1.15,3.6.4.13 Q5SBG8 25286855 407 GTENLYFQSNADTGCAIDISRQELRCGSGVFIHNDVEAWMDRYKYYPETPQGLAKIIQKAHKEGVCGLRSVSRLEHQMWEAVKDELNTLLKENGVDLSVVVEKQEGMYKSAPKRLTATANNTFVVDGPETKECPTQNRAWNSLEVEDFGFGLTSTRMFLKVRESNTTECDSKIIGTAVKNNLAIHSDLSYWIESRLNDTWKLERAVLGEVKSCTWPETHTLWGDGILESDLIIPVTLAGPRSNHNRRPGYKTQNQGPWDEGRVEIDFDYCPGTTVTLSESCGHRGPATRTTTESGKLITDWCCRSCTLPPLRYQTDSGCWYGMEIRPQRHDEKTLVQSQVNA 6z1w A 2.48 BS01 OXN A 1 W36 Q90 S107 Q108 W31 Q85 S102 Q103 1.1.1.n12,4.2.1.107,4.2.1.119 P51659 201 LQSTFVFEEIGRRLKDIGPEVVKKVNAVFEWHITKGGNIGAKWTIDLKSGSGKVYQGPAKGAADTTIILSDEDFMEVVLGKLDPQKAFFSGRLKCRGNIMLSQKLQMILKDYAKL 6z1x A 2.09 BS01 OXN A 1 W36 Q90 M105 S107 Q108 Q111 W31 Q85 M100 S102 Q103 Q106 1.1.1.n12,4.2.1.107,4.2.1.119 P51659 201 LQSTFVFEEIGRRLKDIGPEVVKKVNAVFEWHITKGGNIGAKWTIDLKSGSGKVYQGPAKGAADTTIILSDEDFMEVCLGKLDPQKAFFSGRLKARGNIMLSQKLQMILKDYAKL 7vud A 2.8 BS01 OXN A 1 F98 E189 Y238 F336 D401 F526 F93 E184 Y233 F331 D396 F521 1.14.99.n4 0009570,0010436,0016121,0016702,0046872,0051213 D4QE74 601 DAQRTGNIVAVKPKPSQGLTSKAIDWLEWLFVKMMHDSKQPLHYLSGNFAPVDETPPLKDLPVTGHLPECLNGEFVRVGPNPKFASIAGYHWFDGDGMIHGMRIKDGKATYVSRYVQTSRLKQEEFFGRAMFMKIGDLKGMFGLLMVNMQMLRAKLKVLDISYGIGTANTALVYHHGKLLALSEADKPYAIKVLEDGDLQTIGLLDYDKRLAHSFTAHPKVDPFTGEMFTFGYSHTPPYVTYRVISKDGAMNDPVPITVSGPIMMHDFAITENYAIFMDLPLYFKPKEMVKDKKFIFSFDATQKARFGILPRYAKNELLIKWFELPNCFIFHNANAWEEGDEVVLITCRLENPDLDMVNSTVKERLDNFKNELYEMRFNLQNGLASQKKLSVSAVDFPRVNESYTTRKQRYVYGTTLDKIAKVTGIIKFDLHAEPETGKEKLELGGNVKGIFDLGPGRFGSEAVFVPRHPGITSEEDDGYLIFFVHDENTGKSAVNVIDAKTMSPDPVAVVELPKRVPYGFHAFFVTEDQLQEQA 7vud A 2.8 BS02 OXN A 2 K326 W327 Q386 N387 G388 K321 W322 Q381 N382 G383 1.14.99.n4 0009570,0010436,0016121,0016702,0046872,0051213 D4QE74 602 DAQRTGNIVAVKPKPSQGLTSKAIDWLEWLFVKMMHDSKQPLHYLSGNFAPVDETPPLKDLPVTGHLPECLNGEFVRVGPNPKFASIAGYHWFDGDGMIHGMRIKDGKATYVSRYVQTSRLKQEEFFGRAMFMKIGDLKGMFGLLMVNMQMLRAKLKVLDISYGIGTANTALVYHHGKLLALSEADKPYAIKVLEDGDLQTIGLLDYDKRLAHSFTAHPKVDPFTGEMFTFGYSHTPPYVTYRVISKDGAMNDPVPITVSGPIMMHDFAITENYAIFMDLPLYFKPKEMVKDKKFIFSFDATQKARFGILPRYAKNELLIKWFELPNCFIFHNANAWEEGDEVVLITCRLENPDLDMVNSTVKERLDNFKNELYEMRFNLQNGLASQKKLSVSAVDFPRVNESYTTRKQRYVYGTTLDKIAKVTGIIKFDLHAEPETGKEKLELGGNVKGIFDLGPGRFGSEAVFVPRHPGITSEEDDGYLIFFVHDENTGKSAVNVIDAKTMSPDPVAVVELPKRVPYGFHAFFVTEDQLQEQA 7vud A 2.8 BS03 OXN A 3 S21 L161 S16 L156 1.14.99.n4 0009570,0010436,0016121,0016702,0046872,0051213 D4QE74 603 DAQRTGNIVAVKPKPSQGLTSKAIDWLEWLFVKMMHDSKQPLHYLSGNFAPVDETPPLKDLPVTGHLPECLNGEFVRVGPNPKFASIAGYHWFDGDGMIHGMRIKDGKATYVSRYVQTSRLKQEEFFGRAMFMKIGDLKGMFGLLMVNMQMLRAKLKVLDISYGIGTANTALVYHHGKLLALSEADKPYAIKVLEDGDLQTIGLLDYDKRLAHSFTAHPKVDPFTGEMFTFGYSHTPPYVTYRVISKDGAMNDPVPITVSGPIMMHDFAITENYAIFMDLPLYFKPKEMVKDKKFIFSFDATQKARFGILPRYAKNELLIKWFELPNCFIFHNANAWEEGDEVVLITCRLENPDLDMVNSTVKERLDNFKNELYEMRFNLQNGLASQKKLSVSAVDFPRVNESYTTRKQRYVYGTTLDKIAKVTGIIKFDLHAEPETGKEKLELGGNVKGIFDLGPGRFGSEAVFVPRHPGITSEEDDGYLIFFVHDENTGKSAVNVIDAKTMSPDPVAVVELPKRVPYGFHAFFVTEDQLQEQA