6oyt A 2.824 BS01 NJV A 1 L686 G687 V694 A707 K709 M754 E755 Q756 V757 G759 G760 L810 D822 L21 G22 V29 A42 K44 M84 E85 Q86 V87 G89 G90 L140 D152 D803 K805 D807 N808 D822 D133 K135 D137 N138 D152 2.7.11.25 0004672,0005524,0006468 -logKd/Ki=8.23, IC50=5.9nM IC50=20nM Q99683 31710475 1001 MESDLLEYDYEYDENGDRVVLGKGTYGIVYAGRDLSNQVRIAIKEIPERQPLHEEIALHKHLKHKNIVQYLGSFSENGFIKIFMEQVPGGSLSALLRSKWGPLKDNEQTIGFYTKQILEGLKYLHDNQIVHRDIKGDNVLINTYSGVLKISDFGTSKRLGKAADIWSLGCTIIEMATGKPPVHPEIPESMSAEAKAFILKCFEPDPDKRACANDLLVDEFLK 6oyt B 2.824 BS01 NJV B 1 L686 V694 A707 K709 E755 Q756 V757 P758 G759 L810 D822 L17 V25 A38 K40 E80 Q81 V82 P83 G84 L135 D147 D803 K805 D807 N808 D822 T842 D128 K130 D132 N133 D147 T157 2.7.11.25 0004672,0005524,0006468 IC50=20nM Q99683 31710475 1001 LLEYDYEYDENGDRVVLGKGTYGIVYAGRDLSNQVRIAIKEIPSQPLHEEIALHKHLKHKNIVQYLGSFSENGFIKIFMEQVPGGSLSALLRSKWGPLKDNEQTIGFYTKQILEGLKYLHDNQIVHRDIKGDNVLINTYSGVLKISDFGTSKRLAGTLQYMAPEIGKAADIWSLGCTIIEMATGKPPAAMFKVGMFKVHPEIPESMSAEAKAFILKCFEPDPDKRACANDLLVDEFLK 6oyt C 2.824 BS01 NJV C 1 L686 G687 V694 A707 K709 M754 E755 Q756 V757 P758 G759 L810 D822 L16 G17 V24 A37 K39 M84 E85 Q86 V87 P88 G89 L140 D152 D803 K805 D807 N808 D822 D133 K135 D137 N138 D152 2.7.11.25 0004672,0005524,0006468 -logKd/Ki=8.23, IC50=5.9nM IC50=20nM Q99683 31710475 1001 LEYDYEYDENGDRVVLGKGTYGIVYAGRDLSNQVRIAIKEIPERDSRYSQPLHEEIALHKHLKHKNIVQYLGSFSENGFIKIFMEQVPGGSLSALLRSKWGPLKDNEQTIGFYTKQILEGLKYLHDNQIVHRDIKGDNVLINTYSGVLKISDFGTSKRLLQYMAPEIIDKGPRGGKAADIWSLGCTIIEMATGKPPFHPEIPESMSAEAKAFILKCFEPDPDKRACANDLLVDEFL 6oyt D 2.824 BS01 NJV D 1 L686 G687 V694 A707 K709 M754 E755 Q756 V757 P758 G759 L810 D822 L21 G22 V29 A42 K44 M85 E86 Q87 V88 P89 G90 L141 D153 D803 K805 D807 N808 D822 T842 D134 K136 D138 N139 D153 T163 2.7.11.25 0004672,0005524,0006468 IC50=20nM Q99683 31710475 1002 MESDLLEYDYEYDENGDRVVLGKGTYGIVYAGRDLSNQVRIAIKEIPERSQPLHEEIALHKHLKHKNIVQYLGSFSENGFIKIFMEQVPGGSLSALLRSKWGPLKDNEQTIGFYTKQILEGLKYLHDNQIVHRDIKGDNVLINTYSGVLKISDFGTSKRLAGTLQYMAPEIIYGKAADIWSLGCTIIEMATGKPPFYEPQAAMFKVGMFKVHPEIPESMSAEAKAFILKCFEPDPDKRACANDLLVDEFLKHH