1c6y A 2.5 BS01 MK1 B 1 D25 G48 G49 I50 T82 D25 G48 G49 I50 T82 3.4.24.- 0004190,0006508 -logKd/Ki=9.51, Ki=0.31nM O09893 10739910 524 PQITLWQRPVVTIKIGGQLMEALIDTGADDTVLEEMDLPGRWKPKIIGGIGGFVKVRQYDQIPIEICGHKVIGTVLVGPTPTNIIGRNLLTQIGCTLNF 1c6y B 2.5 BS01 MK1 B 1 D225 G227 A228 D229 D230 V232 G248 P281 I284 D25 G27 A28 D29 D30 V32 G48 P81 I84 D225 T226 G227 D25 T26 G27 3.4.24.- 0004190,0006508 Ki=0.31nM -logKd/Ki=9.51, Ki=0.31nM O09893 10739910 524 PQITLWQRPVVTIKIGGQLMEALIDTGADDTVLEEMDLPGRWKPKIIGGIGGFVKVRQYDQIPIEICGHKVIGTVLVGPTPTNIIGRNLLTQIGCTLNF 1hsg A 2.0 BS01 MK1 B 1 R8 D25 G27 G48 G49 V82 R8 D25 G27 G48 G49 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 -logKd/Ki=9.42, Ki=0.38nM P03367 7929352 902 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hsg B 2.0 BS01 MK1 B 1 D25 G27 A28 D29 D30 V32 I47 G48 I50 P81 D25 G27 A28 D29 D30 V32 I47 G48 I50 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.38nM -logKd/Ki=9.42, Ki=0.38nM P03367 7929352 902 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 1hsh A 1.9 BS01 MK1 A 1 D25 G27 A28 D29 D30 I32 V47 G48 P81 D25 G27 A28 D29 D30 I32 V47 G48 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.47 0004190,0006508 Ki=2.45nM -logKd/Ki=9.42, Ki=0.38nM P04584 7929352 401 PQFSLWKRPVVTAYIEGQPVEVLLDTGADDSIVAGIELGNNYSPKIVGGIGGFINTKEYKNVEIEVLNKKVRATIMTGDTPINIFGRNILTALGMSLNL 1hsh B 1.9 BS01 MK1 A 1 D25 G27 V47 G48 G49 I82 D25 G27 V47 G48 G49 I82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.47 0004190,0006508 -logKd/Ki=9.42, Ki=0.38nM P04584 7929352 401 PQFSLWKRPVVTAYIEGQPVEVLLDTGADDSIVAGIELGNNYSPKIVGGIGGFINTKEYKNVEIEVLNKKVRATIMTGDTPINIFGRNILTALGMSLNL 1hsh C 1.9 BS01 MK1 C 1 D25 G27 A28 D29 D30 I32 G48 I50 P81 I82 D25 G27 A28 D29 D30 I32 G48 I50 P81 I82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.47 0004190,0006508 Ki=2.45nM P04584 7929352 402 PQFSLWKRPVVTAYIEGQPVEVLLDTGADDSIVAGIELGNNYSPKIVGGIGGFINTKEYKNVEIEVLNKKVRATIMTGDTPINIFGRNILTALGMSLNL 1hsh D 1.9 BS01 MK1 C 1 D25 G27 G48 G49 I82 D25 G27 G48 G49 I82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.47 0004190,0006508 P04584 7929352 402 PQFSLWKRPVVTAYIEGQPVEVLLDTGADDSIVAGIELGNNYSPKIVGGIGGFINTKEYKNVEIEVLNKKVRATIMTGDTPINIFGRNILTALGMSLNL 1k6c A 2.2 BS01 MK1 B 1 R8 D25 G27 G48 R8 D25 G27 G48 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 -logKd/Ki=7.48, Kd=33nM P35963 11790852 902 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 1k6c B 2.2 BS01 MK1 B 1 D25 G27 A28 D29 D30 G48 P81 D25 G27 A28 D29 D30 G48 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Kd=33nM -logKd/Ki=7.48, Kd=33nM P35963 11790852 902 PQITLWKRPLVTIRIGGQLKEALLDTGADDTVLEEMNLPGRWKPKMIGGIGGFIKVRQYDQIPIEICGHKAIGTVLVGPTPTNVIGRNLLTQIGCTLNF 1sdt A 1.3 BS01 MK1 B 1 R8 D25 G27 G48 G49 I50 V82 I84 R8 D25 G27 G48 G49 I50 V82 I84 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 -logKd/Ki=9.27, Ki=540pM P03367 15066177 902 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1sdt B 1.3 BS01 MK1 B 1 D125 G127 A128 D129 D130 G148 G149 P181 V182 D25 G27 A28 D29 D30 G48 G49 P81 V82 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=540pM -logKd/Ki=9.27, Ki=540pM P03367 15066177 902 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 1sdu A 1.25 BS01 MK1 B 1 R8 D25 G27 G48 G49 V82 R8 D25 G27 G48 G49 V82 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 -logKd/Ki=10.07, Ki=86pM P03367 15066177 902 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLMTQIGATLNF 1sdu B 1.25 BS01 MK1 B 1 R108 D125 G127 A128 D129 D130 I147 G148 P181 R8 D25 G27 A28 D29 D30 I47 G48 P81 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=86pM -logKd/Ki=10.07, Ki=86pM P03367 15066177 902 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLMTQIGATLNF 1sdv A 1.4 BS01 MK1 B 1 D25 G27 G48 G49 I50 I84 D25 G27 G48 G49 I50 I84 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 -logKd/Ki=8.74, Ki=1810pM P03367 15066177 902 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPANIIGRNLLTQIGATLNF 1sdv B 1.4 BS01 MK1 B 1 D125 G127 A128 D129 D130 I147 G148 G149 I150 P181 D25 G27 A28 D29 D30 I47 G48 G49 I50 P81 D125 T126 G127 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=1810pM -logKd/Ki=8.74, Ki=1810pM P03367 15066177 902 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPANIIGRNLLTQIGATLNF 1sgu A 1.9 BS01 MK1 B 1 D25 G27 I47 G48 I50 P81 A82 D25 G27 I47 G48 I50 P81 A82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 -logKd/Ki=5.37, Ki=4235nM P03367 15379553 2632 PQITLWQRPLVTIKIGGQLREALLDTGADDTIFEEISLPGRWKPKMIGGIGGFVKVRQYDQIPIEICGHKVIGTVLVGPTPANVIGRNLMTQIGCTLNF 1sgu B 1.9 BS01 MK1 B 1 R8 D25 G27 A28 D29 D30 I32 I47 I50 P81 R8 D25 G27 A28 D29 D30 I32 I47 I50 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=4235nM -logKd/Ki=5.37, Ki=4235nM P03367 15379553 2632 PQITLWQRPLVTIKIGGQLREALLDTGADDTIFEEISLPGRWKPKMIGGIGGFVKVRQYDQIPIEICGHKVIGTVLVGPTPANVIGRNLMTQIGCTLNF 2avo A 1.1 BS01 MK1 B 1 R8 D25 G48 G49 V82 I84 R8 D25 G48 G49 V82 I84 D25 T26 G27 D25 T26 G27 3.4.23.16 0004190,0006508,0042802 -logKd/Ki=8.85, Ki=1.40nM Q7SSI0 16277992 902 PQITLWKRPLVTIKIGGQLKEALIDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2avo B 1.1 BS01 MK1 B 1 D25 G27 A28 D29 D30 V32 I47 G48 G49 P81 V82 D25 G27 A28 D29 D30 V32 I47 G48 G49 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508,0042802 Ki=1.4nM -logKd/Ki=8.85, Ki=1.40nM P04587 16277992 902 PQITLWKRPLVTIKIGGQLKEALIDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2avs A 1.1 BS01 MK1 B 1 R8 D25 G27 G48 G49 P81 V82 I84 R8 D25 G27 G48 G49 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 -logKd/Ki=7.57, Ki=27.0nM P04587 16277992 902 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGVGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2avs B 1.1 BS01 MK1 B 1 R8 D25 G27 A28 D29 D30 V32 G48 G49 P81 V82 R8 D25 G27 A28 D29 D30 V32 G48 G49 P81 V82 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=27nM -logKd/Ki=7.57, Ki=27.0nM P04587 16277992 902 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGVGGFIKVRQYDQIIIEIAGHKAIGTVLVGPTPVNIIGRNLLTQIGATLNF 2avv A 1.5 BS01 MK1 A 1 R8 D25 G27 A28 G48 G49 V82 I84 R8 D25 G27 A28 G48 G49 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.55nM -logKd/Ki=9.26, Ki=0.55nM P04587 16277992 901 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAISTVLVGPTPVNIIGRNLLTQIGATLNF 2avv B 1.5 BS01 MK1 A 1 D25 G27 A28 D29 D30 V32 I47 G48 I50 P81 I84 D25 G27 A28 D29 D30 V32 I47 G48 I50 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 -logKd/Ki=9.26, Ki=0.55nM P04587 16277992 901 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAISTVLVGPTPVNIIGRNLLTQIGATLNF 2avv D 1.5 BS01 MK1 E 1 R8 D25 G27 G48 G49 V82 I84 R8 D25 G27 G48 G49 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 P04587 16277992 902 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAISTVLVGPTPVNIIGRNLLTQIGATLNF 2avv E 1.5 BS01 MK1 E 1 D25 G27 A28 D29 D30 G48 I50 P81 I84 D25 G27 A28 D29 D30 G48 I50 P81 I84 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=0.55nM P04587 16277992 902 PQITLWKRPLVTIKIGGQLKEALLDTGADDTVIEEMSLPGRWKPKMIGGIGGFIKVRQYDQIIIEIAGHKAISTVLVGPTPVNIIGRNLLTQIGATLNF 2b7z A 2.2 BS01 MK1 B 1 R8 D25 G27 I47 G48 G49 I50 R8 D25 G27 I47 G48 G49 I50 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 P03367 200 PQITLWQRPLVTIKIGGQLREALLDTGADDTIFEEISLPGRWKPKIIGGIGGFIKVRQYDQIPIEICGHKVIGTVLVGPTPANVIGRNLMTQIGCTLNF 2b7z B 2.2 BS01 MK1 B 1 D25 G27 D29 D30 I32 I47 I50 P81 D25 G27 D29 D30 I32 I47 I50 P81 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 P03367 200 PQITLWQRPLVTIKIGGQLREALLDTGADDTIFEEISLPGRWKPKIIGGIGGFIKVRQYDQIPIEICGHKVIGTVLVGPTPANVIGRNLMTQIGCTLNF 2bpx A 2.8 BS01 MK1 B 1 R8 D25 G27 G48 V82 I84 R8 D25 G27 G48 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 -logKd/Ki=9.40, Ki=0.4nM P04587 9757136 902 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2bpx B 2.8 BS01 MK1 B 1 D25 G27 A28 D29 D30 V32 I47 P81 I84 D25 G27 A28 D29 D30 V32 I47 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 -logKd/Ki=9.40, Ki=0.4nM P04587 9757136 902 PQITLWQRPLVTIKIGGQLKEALLDTGADDTVLEEMSLPGRWKPKMIGGIGGFIKVRQYDQILIEICGHKAIGTVLVGPTPVNIIGRNLLTQIGCTLNF 2r5p A 2.3 BS01 MK1 B 1 R8 D25 G27 G48 G49 I50 V82 I84 R8 D25 G27 G48 G49 I50 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 -logKd/Ki=8.48, Ki=3.3nM O12158 18092815 902 PQITLWKRPLVSIKVGGQIKEALLDTGADDTVIEEIALPGRWKPKMIGGIGGFIKVRQYDQIIIEICGKKAIGTVLVGPTPVNIIGRNMLTQLGCTLNF 2r5p B 2.3 BS01 MK1 B 1 D25 G27 A28 D29 D30 V32 G48 G49 P81 V82 I84 D25 G27 A28 D29 D30 V32 G48 G49 P81 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=3.3nM -logKd/Ki=8.48, Ki=3.3nM O12158 18092815 902 PQITLWKRPLVSIKVGGQIKEALLDTGADDTVIEEIALPGRWKPKMIGGIGGFIKVRQYDQIIIEICGKKAIGTVLVGPTPVNIIGRNMLTQLGCTLNF 2r5p C 2.3 BS01 MK1 D 1 R8 D25 G27 G48 G49 I50 V82 I84 R8 D25 G27 G48 G49 I50 V82 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 O12158 18092815 902 PQITLWKRPLVSIKVGGQIKEALLDTGADDTVIEEIALPGRWKPKMIGGIGGFIKVRQYDQIIIEICGKKAIGTVLVGPTPVNIIGRNMLTQLGCTLNF 2r5p D 2.3 BS01 MK1 D 1 D25 G27 A28 D29 D30 G48 G49 P81 I84 D25 G27 A28 D29 D30 G48 G49 P81 I84 D25 T26 G27 D25 T26 G27 2.7.7.-,2.7.7.49,2.7.7.7,3.1.-.-,3.1.13.2,3.1.26.13,3.4.23.16 0004190,0006508 Ki=3.3nM O12158 18092815 902 PQITLWKRPLVSIKVGGQIKEALLDTGADDTVIEEIALPGRWKPKMIGGIGGFIKVRQYDQIIIEICGKKAIGTVLVGPTPVNIIGRNMLTQLGCTLNF 3wsj A 2.404 BS01 MK1 A 1 R10 D32 G34 D36 M37 V39 L91 W98 R10 D32 G34 D36 M37 V39 L91 W98 ? 0004190,0006508,0008233,0046872 Ki=35uM Q82134 25006983 201 PVIPLDPARRPVIKAQVDTQTSHPKTIEALLDTGADMTVIPIALFSSNTPLKNTSVLGAGGQTQDHFKLTSLPVLIRLPFRTTPIVLTSCLVDTKNNWAIIGRDALQQCQGVLYLP 3wsj B 2.404 BS01 MK1 A 1 R10 D32 G34 W98 R10 D32 G34 W98 ? 0004190,0006508,0008233,0046872 Q82134 25006983 201 PVIPLDPARRPVIKAQVDTQTSHPKTIEALLDTGADMTVIPIALFSSNTPLKNTSVLGAGGQTQDHFKLTSLPVLIRLPFRTTPIVLTSCLVDTKNNWAIIGRDALQQCQGVLYLP