1w7g H 1.65 BS03 MIU H 1 H57 Y60A W60D K60F A190 C191 E192 W215 G216 G219 H43 Y47 W50 K52 A194 C195 E196 W221 G222 G224 3.4.21.5 0004252,0005509,0006508,0007596 Ki~13uM -logKd/Ki=5.10, Ki=8uM Ki=1900nM P00734 16294249 300 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETWGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQFG