1dwd H 3.0 BS03 MID H 1 H57 Y60A W60D N98 L99 I174 D189 A190 W215 G216 H43 Y47 W50 N95 L96 I179 D199 A200 W227 G228 3.4.21.5 0004252,0005509,0006508,0007596 -logKd/Ki=8.18, Ki=6.6nM Ki=6nM, IC50=690nM, EC50=750nM P00734 1939071 1 IVEGSDAEIGMSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTENDLLVRIGKHSRTRYERNIEKISMLEKIYIHPRYNWRENLDRDIALMKLKKPVAFSDYIHPVCLPDRETAASLLQAGYKGRVTGWGNLKETWTANVGKGQPSVLQVVNLPIVERPVCKDSTRIRITDNMFCAGYKPDEGKRGDACEGDSGGPFVMKSPFNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDQF 1ets H 2.3 BS01 MID H 1 H57 W60D N98 L99 D189 A190 E192 S195 W215 G216 E217 G219 C220 H43 W50 N95 L96 D199 A200 E202 S205 W227 G228 E229 G230 C231 3.4.21.5 0004252,0005509,0006508,0007596 Ki=6nM -logKd/Ki=8.22, Ki=6nM Ki=6nM P00735 1518046 1 IVEGQDAEVGLSPWQVMLFRKSPQELLCGASLISDRWVLTAAHCLLYPPWDKNFTVDDLLVRIGKHSRTRYERKVEKISMLDKIYIHPRYNWKENLDRDIALLKLKRPIELSDYIHPVCLPDKQTAAKLLHAGFKGRVTGWGNRRETWTTSVAEVQPSVLQVVNLPLVERPVCKASTRIRITDNMFCAGYKPGEGKRGDACEGDSGGPFVMKSPYNNRWYQMGIVSWGEGCDRDGKYGFYTHVFRLKKWIQKVIDRLGS 1ppc E 1.8 BS01 MID E 1 H57 N97 L99 D189 S190 S195 W215 G216 G219 H40 N79 L81 D171 S172 S177 W193 G194 G196 G193 S195 G196 G175 S177 G178 3.4.21.4 0004175,0004252,0005515,0005576,0005615,0006508,0007586,0008236,0046872,0097180,0097655 Ki=0.69uM -logKd/Ki=6.16, Ki=0.69uM Ki=325nM P00760 2226434 5 IVGGYTCGANTVPYQVSLNSGYHFCGGSLINSQWVVSAAHCYKSGIQVRLGEDNINVVEGNEQFISASKSIVHPSYNSNTLNNDIMLIKLKSAASLNSRVASISLPTSCASAGTQCLISGWGNTKSSGTSYPDVLKCLKAPILSDSSCKSAYPGQITSNMFCAGYLEGGKDSCQGDSGGPVVCSGKLQGIVSWGSGCAQKNKPGVYTKVCNYVSWIKQTIASN