3eyg	A	1.9	BS01	MI1	A	1	L881 G882 E883 G884 G887 V889 A906 K908 M956 F958 L959 L1010 G1020 D1021	L17 G18 E19 G20 G23 V25 A42 K44 M84 F86 L87 L138 G148 D149	D1003 A1005 R1007 N1008 D1021 D1040	D131 A133 R135 N136 D149 D168	2.7.10.2	0004672,0004713,0005524,0006468		ic50=1.6nM	-logKd/Ki=8.80, IC50=1.6nM	IC50=15nM, EC50=53nM, Kd=>10000nM, Ki=0.700000nM	P23458	19361440	1 	VDPTHFEKRFLKRIRDLGEGHFGKVELCRYDPEGDNTGEQVAVKSLKPHIADLKKEIEILRNLYHENIVKYKGICTENGIKLIMEFLPSGSLKEYLPKNKNKINLKQQLKYAVQICKGMDYLGSRQYVHRDLAARNVLVESEHQVKIGDFGLTKAIETDKEYYTVKDDRDSPVFWYAPECLMQSKFYIASDVWSFGVTLHELLTYCDSDSSPMALFLKMIGPTHGQMTVTRLVNTLKEGKRLPCPPNCPDEVYQLMRKCWEFQPSNRTSFQNLIEGFEALLK
3fup	A	2.4	BS01	MI1	A	1	L855 G856 K857 G858 G861 V863 A880 Y931 L932 L983 G993 D994	L13 G14 K15 G16 G19 V21 A38 Y85 L86 L137 G147 D148	D976 A978 R980 N981 D994 S1016	D130 A132 R134 N135 D148 S170	2.7.10.2	0004672,0004713,0005524,0006468		ic50=21.7nM	-logKd/Ki=7.66, IC50=21.7nM	IC50=77nM, EC50=93nM, Kd=5nM, Ki=0.700000nM	O60674	19361440	1 	QFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDQMAG
3fup	B	2.4	BS01	MI1	B	1	G856 K857 G858 G861 S862 V863 A880 M929 Y931 L932 L983 G993 D994	G17 K18 G19 G22 S23 V24 A41 M86 Y88 L89 L140 G150 D151	D976 A978 R980 N981 D994 S1016	D133 A135 R137 N138 D151 S173	2.7.10.2	0004672,0004713,0005524,0006468		ic50=21.7nM		IC50=77nM, EC50=93nM, Kd=5nM, Ki=0.700000nM	O60674	19361440	1 	DPTQFEERHLKFLQQLGKGNFGSVEMCRYDPLQDNTGEVVAVKKLQHSTEEHLRDFEREIEILKSLQHDNIVKYKGVCYSNLKLIMEYLPYGSLRDYLQKHKERIDHIKLLQYTSQICKGMEYLGTKRYIHRDLATRNILVENENRVKIGDFGLTKVLPQDKEYYKVKEPGESPIFWYAPESLTESKFSVASDVWSFGVVLYELFTYIEKSKSPPAEFMRMIGNDKQGQMIVFHLIELLKNNGRLPRPDGCPDEIYMIMTECWNNNVNQRPSFRDLALRVDQIRDQMAG
3lxk	A	2.0	BS01	MI1	A	1	G829 K830 G831 G834 S835 V836 A853 Y904 L905 R953 L956 D967	G15 K16 G17 G20 S21 V22 A39 Y90 L91 R139 L142 D153	D949 A951 R953 N954 D967	D135 A137 R139 N140 D153	2.7.10.2	0004672,0004713,0005524,0006468		Ki=0.2nM	-logKd/Ki=9.80, Kd=0.16nM	IC50=55nM, Ki=0.400000nM, Kd=2.2nM	P52333	20478313	1125 	TIFEERHLKYISQLGKGNFGSVELCRYDPLGDNTGALVAVKQLQHSGPDQQRDFQREIQILKALHSDFIVKYRGVSYGPGRQSLRLVMEYLPSGCLRDFLQRHRARLDASRLLLYSSQICKGMEYLGSRRCVHRDLAARNILVESEAHVKIADFGLAKLLPLDKDYYVVREPGQSPIFWYAPESLSDNIFSRQSDVWSFGVVLYELFTYCDKSCSPSAEFLRMMVPALSRLLELLEEGQRLPAPPACPAEVHELMKLCWAPSPQDRPSFSALGPQLDML
3lxn	A	2.5	BS01	MI1	A	1	L903 G904 E905 G906 G909 V911 A928 K930 I960 E979 Y980 V981 L1030 G1040 D1041	L16 G17 E18 G19 G22 V24 A41 K43 I73 E92 Y93 V94 L143 G153 D154	D1023 A1025 R1027 N1028 D1041 P1064	D136 A138 R140 N141 D154 P174	2.7.10.2	0004672,0004713,0005524,0006468		Ki=4.4nM		IC50=489nM, Kd=620nM, Ki=4.39nM	P29597	20478313	1 	DPTVFHKRYLKKIRDLGEGHFGKVSLYCYDPTNDGTGEMVAVKALKADAGPQHRSGWKQEIDILRTLYHEHIIKYKGCCEDAGAASLQLVMEYVPLGSLRDYLPRHSIGLAQLLLFAQQICEGMAYLHAQHYIHRDLAARNVLLDNDRLVKIGDFGLAKAVPEGHEYYRVGDSPVFWYAPECLKEYKFYYASDVWSFGVTLYELLTHCDSSQSPPTKFLELIGIAQGQMTVLRLTELLERGERLPRPDKCPAEVYHLMKNCWETEASFRPTFENLIPILKTVHEKYQG
4oti	A	1.93	BS01	MI1	A	1	G628 R629 G630 G633 V635 A648 S704 L753 F910	G17 R18 G19 G22 V24 A37 S93 L142 F268	D746 K748 D750 N751 D764	D135 K137 D139 N140 D153	2.7.11.13	0004672,0004674,0005524,0006468		ic50=43nM	-logKd/Ki=7.37, IC50=43nM	Kd=200nM	Q16512	25111382	1001 	RKSPLTLEDFKFLAVLGRGHFGKVLLSEFRPSGELFAIKALKKGDIVARDEVESLMCEKRILAAVTSAGHPFLVNLFGCFQTPEHVCFVMEYSAGGDLMLHIHSDVFSEPRAIFYSACVVLGLQFLHEHKIVYRDLKLDNLLLDTEGYVKIADFGLTRAVDWWGLGVLLYEMLVGESPFPGDDEEEVFDSIVNDEVRYPRFLSAEAIGIMRRLLRRNPERRLGSSERDAEDVKKQPFFRTLGWEALLARRLPPPFVPTLSGRTDVSNFDEEFTGEAPTLSPPRDARPLTAAEQAAFLDFDFVAG