3iw4	A	2.8	BS01	LW4	A	1	L345 F350 V353 A366 T401 M417 E418 Y419 V420 D467 M470 A480 D481	L15 F20 V23 A36 T71 M87 E88 Y89 V90 D137 M140 A150 D151	D463 K465 N468 D481 T501	D133 K135 N138 D151 T171	2.7.11.13	0004672,0004674,0004697,0005524,0006468			-logKd/Ki=8.68, IC50=2.1nM	IC50=2.1nM	P17252	19827831	901 	LDRVKLTDFNFLMVLGKGSFGKVMLADRKGTEELYAIKILKKDVVIQDDDVECTMVEKRVLALLDKPPFLTQLHSCFQTVDRLYFVMEYVNGGDLMYHIQQVGKFKEPQAVFYAAEISIGLFFLHKRGIIYRDLKLDNVMLDSEGHIKIADFGMCKEHMMDGVTTREFCGTPDYIAPEIIAYQPYGKSVDWWAYGVLLYEMLAGQPPFDGEDEDELFQSIMEHNVSYPKSLSKEAVSICKGLMTKHPAKRLGCGPEGERDVREHAFFRRIDWEKLENREIQPPFKPKVFDKFFTRGQPVLTPPDQLVIANIDQSDFEGFSYVNPQFVHPILQ
3iw4	B	2.8	BS01	LW4	B	1	L345 F350 V353 A366 T401 M417 E418 Y419 D467 M470 A480 D481	L14 F19 V22 A35 T70 M86 E87 Y88 D136 M139 A149 D150	D463 K465 N468 D481 T501	D132 K134 N137 D150 T169	2.7.11.13	0004672,0004674,0004697,0005524,0006468				IC50=2.1nM	P17252	19827831	901 	DRVKLTDFNFLMVLGKGSFGKVMLADRKGTEELYAIKILKKDVVIQDDDVECTMVEKRVLALLDKPPFLTQLHSCFQTVDRLYFVMEYVNGGDLMYHIQQVGKFKEPQAVFYAAEISIGLFFLHKRGIIYRDLKLDNVMLDSEGHIKIADFGMCKEHMMGVTTREFCGTPDYIAPEIIAYQPYGKSVDWWAYGVLLYEMLAGQPPFDGEDEDELFQSIMEHNVSYPKSLSKEAVSICKGLMTKHPAKRLGCGPEGERDVREHAFFRRIDWEKLENREIQPPFKPKVFDKFFTRGQPVLTPPDQLVIANIDQSDFEGFSYVNPQFVHP
3iw4	C	2.8	BS01	LW4	C	1	L345 G346 F350 V353 A366 T401 E418 Y419 V420 D467 M470 A480 D481	L16 G17 F21 V24 A37 T72 E89 Y90 V91 D138 M141 A151 D152	D463 K465 N468 D481 T501	D134 K136 N139 D152 T172	2.7.11.13	0004672,0004674,0004697,0005524,0006468				IC50=2.1nM	P17252	19827831	901 	NLDRVKLTDFNFLMVLGKGSFGKVMLADRKGTEELYAIKILKKDVVIQDDDVECTMVEKRVLALLDKPPFLTQLHSCFQTVDRLYFVMEYVNGGDLMYHIQQVGKFKEPQAVFYAAEISIGLFFLHKRGIIYRDLKLDNVMLDSEGHIKIADFGMCKEHMMDGVTTREFCGTPDYIAPEIIAYQPYGKSVDWWAYGVLLYEMLAGQPPFDGEDEDELFQSIMEHNVSYPKSLSKEAVSICKGLMTKHPAKRLGCGPEGERDVREHAFFRRIDWEKLENREIQPPFKPKVFDKFFTRGQPVLTPPDQLVIANIDQSDFEGFSYVNPQFVHPILQS