2w71 A 1.99 BS01 L23 A 1 K159 Y203 L204 H209 Q233 H236 L278 I437 K159 Y203 L204 H209 Q233 H236 L278 I437 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 E296 R338 6.3.4.14 0003824,0003989,0004075,0005515,0005524,0005737,0005829,0006633,0009317,0016874,0042803,0045717,0046872,2001295 ic50=0.334uM -logKd/Ki=6.48, IC50=0.334uM IC50=334nM P24182 19413326 1448 MLDKIVIANRGEIALRILRACKELGIKTVAVHSSADRDLKHVLLADETVCIGPAPSVKSYLNIPAIISAAEITGAVAIHPGYGFLSENANFAEQVERSGFIFIGPKAETIRLMGDKVSAIAAMKKAGVPCVPGSDGPLGDDMDKNRAIAKRIGYPVIIKASGGGGGRGMRVVRGDAELAQSISMTRAEAKAAFSNDMVYMEKYLENPRHVEIQVLADGQGNAIYLAERDCSMQRRHQKVVEEAPAPGITPELRRYIGERCAKACVDIGYRGAGTFEFLFENGEFYFIEMNTRIQVEHPVTEMITGVDLIKEQLRIAAGQPLSIKQEEVHVRGHAVECRINAEDPNTFLPSPGKITRFHAPGGFGVRWESHIYAGYTVPPYYDSMIGKLICYGENRDVAIARMKNALQELIIDGIKTNVDLQIRIMNDENFQHGGTNIHYLEKKLGL 2w71 C 1.99 BS01 L23 C 1 K159 M169 E201 K202 Y203 L204 H209 Q233 H236 L278 I287 I437 K159 M169 E201 K202 Y203 L204 H209 Q233 H236 L278 I287 I437 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 R338 K116 K159 D196 H209 R235 T274 E276 E288 N290 R292 R338 6.3.4.14 0003824,0003989,0004075,0005515,0005524,0005737,0005829,0006633,0009317,0016874,0042803,0045717,0046872,2001295 ic50=0.334uM IC50=334nM P24182 19413326 1448 MLDKIVIANRGEIALRILRACKELGIKTVAVHSSADRDLKHVLLADETVCIGPAPSVKSYLNIPAIISAAEITGAVAIHPGYGFLSENANFAEQVERSGFIFIGPKAETIRLMGDKVSAIAAMKKAGVPCVPGSDGPLGDDMDKNRAIAKRIGYPVIIKASGGGGGRGMRVVRGDAELAQSISMTRAEAKAAFSNDMVYMEKYLENPRHVEIQVLADGQGNAIYLAERDCSMQRRHQKVVEEAPAPGITPELRRYIGERCAKACVDIGYRGAGTFEFLFENGEFYFIEMNTRIQVEHPVTEMITGVDLIKEQLRIAAGQPLSIKQEEVHVRGHAVECRINAEDPNTFLPSPGKITRFHAPGGFGVRWESHIYAGYTVPPYYDSMIGKLICYGENRDVAIARMKNALQELIIDGIKTNVDLQIRIMNDENFQHGGTNIHYLEKKLGL