1kyn A 3.5 BS01 KTP A 1 H57 A190 F191 K192 S195 G216 K217 H44 A176 F177 K178 S181 G198 K199 H57 D102 K192 G193 D194 S195 G196 H44 D88 K178 G179 D180 S181 G182 3.4.21.20 0002003,0002548,0004252,0005515,0005576,0005615,0005634,0005737,0005764,0005829,0005886,0006468,0006508,0006935,0006955,0008201,0008233,0008236,0010494,0016020,0016485,0019221,0019731,0022617,0030141,0030168,0032496,0035578,0035590,0042119,0042742,0043231,0048018,0050778,0050829,0050830,0050832,0050868,0062023,0070062,0070946,0071222,0089720,0098786,1901731 -logKd/Ki=5.39, IC50=4.1uM IC50=4100nM P08311 11942800 601 IIGGRESRPHSRPYMAYLQIQSPAGQSRCGGFLVREDFVLTAAHCWGSNINVTLGAHNIQRRENTQQHITARRAIRHPQYNQRTIQNDIMLLQLSRRVRRNRNVNPVALPRAQEGLRPGTLCTVAGWGRVSMRRGTDTLREVQLRVQRDRQCLRIFGSYDPRRQICVGDRRERKAAFKGDSGGPLLCNNVAHGIVSYGKSSGVPPEVFTRVSSFLPWIRTTMR 1kyn B 3.5 BS01 KTP B 1 H357 I399 K492 G493 S495 S514 Y515 G516 H44 I85 K178 G179 S181 S196 Y197 G198 H357 D402 K492 G493 D494 S495 G496 H44 D88 K178 G179 D180 S181 G182 3.4.21.20 0002003,0002548,0004252,0005515,0005576,0005615,0005634,0005737,0005764,0005829,0005886,0006468,0006508,0006935,0006955,0008201,0008233,0008236,0010494,0016020,0016485,0019221,0019731,0022617,0030141,0030168,0032496,0035578,0035590,0042119,0042742,0043231,0048018,0050778,0050829,0050830,0050832,0050868,0062023,0070062,0070946,0071222,0089720,0098786,1901731 IC50=4100nM P08311 11942800 701 IIGGRESRPHSRPYMAYLQIQSPAGQSRCGGFLVREDFVLTAAHCWGSNINVTLGAHNIQRRENTQQHITARRAIRHPQYNQRTIQNDIMLLQLSRRVRRNRNVNPVALPRAQEGLRPGTLCTVAGWGRVSMRRGTDTLREVQLRVQRDRQCLRIFGSYDPRRQICVGDRRERKAAFKGDSGGPLLCNNVAHGIVSYGKSSGVPPEVFTRVSSFLPWIRTTMRSF