4jr3 A 2.7 BS01 KJR A 1 L694 V702 A719 K721 T766 M769 G772 R817 L820 D831 L23 V31 A48 K50 T95 M98 G101 R146 L149 D160 D813 A815 R817 N818 D831 G850 D142 A144 R146 N147 D160 G179 2.7.10.1 0004672,0004713,0005524,0006468 -logKd/Ki=6.66, IC50=218nM IC50=218nM P00533 23611691 1001 GEAPNQALLRILKETEFKKIKVLGSGAFGTVYKGLWIPEGEKVKIPVAIKELREATSPKANKEILDEAYVMASVDNPHVCRLLGICLTSTVQLITQLMPFGCLLDYVREHKDNIGSQYLLNWCVQIAKGMNYLEDRRLVHRDLAARNVLVKTPQHVKITDFGLAKLLGAEEKEYHAEGGKVPIKWMALESILHRIYTHQSDVWSYGVTVWELMTFGSKPYDGIPASEISSILEKGERLPQPPICTIDVYMIMVKCWMIDADSRPKFRELIIEFSKMARDPQRYLVIQGDDMDDVVDADEYLIP