3qvi A 2.5 BS01 K95 A 1 H32 A34 S35 W39 L291 H33 A35 S36 W40 L289 H32 S35 N37 W39 S75 D215 T218 H33 S36 N38 W40 S76 D213 T216 3.4.23.39 0004190,0005773,0005775,0006508,0016020,0020020,0044002 Q9Y006 21928835 329 EFDNVELKDLANVLSFGEAKLGDNGQKFNFLFHTASSNVWVPSIKCTSESCESKNHYDSSKSKTYEKDDTPVKLTSKAGTISGIFSKDLVTIGKLSVPYKFIEMTEIVGFEPFYSESDVDGVFGLGWKDLSIGSIDPYIVELKTQNKIEQAVYSIYLPPENKNKGYLTIGGIEERFFDGPLNYEKLNHDLMWQVDLDVHFGNVSSKKANVILDSATSVITVPTEFFNQFVESASVFLSLYVTTCGNTKLPTLEYRSPNKVYTLEPKQYLEPLENIFSALCMLNIVPIDLEKNTFVLGDPFMRKYFTVYDYDNHTVGFALAKNL 3qvi C 2.5 BS01 K95 C 1 H32 A34 S35 W39 L128 M189 H33 A35 S36 W40 L130 M191 H32 S35 N37 W39 S75 D215 T218 H33 S36 N38 W40 S76 D213 T216 3.4.23.39 0004190,0005773,0005775,0006508,0016020,0020020,0044002 Q9Y006 21928835 329 EFDNVELKDLANVLSFGEAKLGDNGQKFNFLFHTASSNVWVPSIKCTSESCESKNHYDSSKSKTYEKDDTPVKLTSKAGTISGIFSKDLVTIGKLSVPYKFIEMTEIVGFEPFYSESDVDGVFGLGWKDLSIGSIDPYIVELKTQNKIEQAVYSIYLPPENKNKGYLTIGGIEERFFDGPLNYEKLNHDLMWQVDLDVHFGNVSSKKANVILDSATSVITVPTEFFNQFVESASVFKVPFLSLYVTTCGNTKLPTLEYRSPNKVYTLEPKQYLEPLENIFSALCMLNIVPIDLEKNTFVLGDPFMRKYFTVYDYDNHTVGFALAKNL 3qvi C 2.5 BS02 K95 C 2 E278A L281 E277 L283 H32 S35 N37 W39 S75 D215 T218 H33 S36 N38 W40 S76 D213 T216 3.4.23.39 0004190,0005773,0005775,0006508,0016020,0020020,0044002 Q9Y006 21928835 330 EFDNVELKDLANVLSFGEAKLGDNGQKFNFLFHTASSNVWVPSIKCTSESCESKNHYDSSKSKTYEKDDTPVKLTSKAGTISGIFSKDLVTIGKLSVPYKFIEMTEIVGFEPFYSESDVDGVFGLGWKDLSIGSIDPYIVELKTQNKIEQAVYSIYLPPENKNKGYLTIGGIEERFFDGPLNYEKLNHDLMWQVDLDVHFGNVSSKKANVILDSATSVITVPTEFFNQFVESASVFKVPFLSLYVTTCGNTKLPTLEYRSPNKVYTLEPKQYLEPLENIFSALCMLNIVPIDLEKNTFVLGDPFMRKYFTVYDYDNHTVGFALAKNL 3qvi D 2.5 BS01 K95 C 1 E278A L281 E277 L283 H32 S35 N37 W39 S75 D215 T218 H33 S36 N38 W40 S76 D213 T216 3.4.23.39 0004190,0005773,0005775,0006508,0016020,0020020,0044002 Q9Y006 21928835 329 EFDNVELKDLANVLSFGEAKLGDNGQKFNFLFHTASSNVWVPSIKCTSESCESKNHYDSSKSKTYEKDDTPVKLTSKAGTISGIFSKDLVTIGKLSVPYKFIEMTEIVGFEPFYSESDVDGVFGLGWKDLSIGSIDPYIVELKTQNKIEQAVYSIYLPPENKNKGYLTIGGIEERFFDGPLNYEKLNHDLMWQVDLDVHFGNVSSKKANVILDSATSVITVPTEFFNQFVESASVFKVPFLSLYVTTCGNTKLPTLEYRSPNKVYTLEPKQYLEPLENIFSALCMLNIVPIDLEKNTFVLGDPFMRKYFTVYDYDNHTVGFALAKNL 3qvi D 2.5 BS02 K95 C 2 H32 A34 S35 W39 L73 M189 H33 A35 S36 W40 L74 M191 H32 S35 N37 W39 S75 D215 T218 H33 S36 N38 W40 S76 D213 T216 3.4.23.39 0004190,0005773,0005775,0006508,0016020,0020020,0044002 Q9Y006 21928835 330 EFDNVELKDLANVLSFGEAKLGDNGQKFNFLFHTASSNVWVPSIKCTSESCESKNHYDSSKSKTYEKDDTPVKLTSKAGTISGIFSKDLVTIGKLSVPYKFIEMTEIVGFEPFYSESDVDGVFGLGWKDLSIGSIDPYIVELKTQNKIEQAVYSIYLPPENKNKGYLTIGGIEERFFDGPLNYEKLNHDLMWQVDLDVHFGNVSSKKANVILDSATSVITVPTEFFNQFVESASVFKVPFLSLYVTTCGNTKLPTLEYRSPNKVYTLEPKQYLEPLENIFSALCMLNIVPIDLEKNTFVLGDPFMRKYFTVYDYDNHTVGFALAKNL 5yid A 2.1 BS01 K95 A 1 D36 G38 Y79 V80 S81 I125 G218 T219 S220 L294 F296 I302 D32 G34 Y75 V76 S77 I121 G214 T215 S216 L290 F292 I298 3.4.23.39 0004190,0006508 Ki=4nM -logKd/Ki=5.40, Ki=4.0uM Q8I6V3 29943906 401 NDNIELVDFQNIMFYGDAEVGDNQQPFTFILDTGSANLWVPSVKCTTAGCLTKHLYDSSKSRTYEKDGTKVEMNYVSGTVSGFFSKDLVTVGNLSLPYKFIEVIDTNGFEPTYTASTFDGILGLGWKDLSIGSVDPIVVELKNQNKIENALFTFYLPVHDKHTGFLTIGGIEERFYEGPLTYEKLNHDLYWQITLDAHVGNIMLEKANCIVDSGTSAITVPTDFLNKMLQNLDVIKVPFLPFYVTLCNNSKLPTFEFTSENGKYTLEPEYYLQHIEDVGPGLCMLNIIGLDFPVPTFILGDPFMRKYFTVFDYDNQSVGIALAKKNL