3kcf	A	2.8	BS01	JZO	A	1	I211 A230 K232 L260 S280 Y282 H283 K337 L340 D351	I41 A60 K62 L90 S110 Y112 H113 K167 L170 D181	D333 K335 N338 D351 T375	D163 K165 N168 D181 T203	2.7.11.30	0004672,0004675,0005524,0006468,0007178,0016020			-logKd/Ki=7.46, Ki=0.035uM	IC50=3690nM, Ki=35nM	P36897	19914068	1 	ISEGTTLKDLIYDMTTSGSGSGLPLLVQRTIARTIVLQESIGKGRFGEVWRGKWRGEEVAVKIFSSREERSWFREAEIYQTVMLRHENILGFIAADNKDNGTWTQLWLVSDYHEHGSLFDYLNRYTVTVEGMIKLALSTASGLAHLHMEIVGTQGKPAIAHRDLKSKNILVKKNGTCCIADLGLAVRHDSATDTIDINHRVGTKRYMAPEVLDDSINMKHFESFKRADIYAMGLVFWEIARRCSIGGIHEDYQLPYYDLVPSDPSVEEMRKVVCEQKLRPNIPNRWQSCEALRVMAKIMRECWYANGAARLTALRIKKTLSQLSQQEG
3kcf	B	2.8	BS01	JZO	B	1	A230 K232 Y249 L260 S280 Y282 H283 L340	A60 K62 Y79 L90 S110 Y112 H113 L166	D333 K335 N338 D351 T375	D159 K161 N164 D177 T198	2.7.11.30	0004672,0004675,0005524,0006468,0007178,0016020				IC50=3690nM, Ki=35nM	P36897	19914068	2 	ISEGTTLKDLIYDMTTSGSGSGLPLLVQRTIARTIVLQESIGKGRFGEVWRGKWRGEEVAVKIFSSREERSWFREAEIYQTVMLRHENILGFIAADNKDNGTWTQLWLVSDYHEHGSLFDYLNRYTVTVEGMIKLALSTASGLAHLHMEIGKPAIAHRDLKSKNILVKKNGTCCIADLGLAVRHDSATDTIDIHRVGTKRYMAPEVLDDSINMKHFESFKRADIYAMGLVFWEIARRCSIGGIHEDYQLPYYDLVPSDPSVEEMRKVVCEQKLRPNIPNRWQSCEALRVMAKIMRECWYANGAARLTALRIKKTLSQLSQQEGI
3kcf	C	2.8	BS01	JZO	C	1	I211 A230 K232 Y249 L260 S280 Y282 H283 L340 D351	I41 A60 K62 Y79 L90 S110 Y112 H113 L170 D181	D333 K335 N338 D351 T375	D163 K165 N168 D181 T205	2.7.11.30	0004672,0004675,0005524,0006468,0007178,0016020				IC50=3690nM, Ki=35nM	P36897	19914068	3 	ISEGTTLKDLIYDMTTSGSGSGLPLLVQRTIARTIVLQESIGKGRFGEVWRGKWRGEEVAVKIFSSREERSWFREAEIYQTVMLRHENILGFIAADNKDNGTWTQLWLVSDYHEHGSLFDYLNRYTVTVEGMIKLALSTASGLAHLHMEIVGTQGKPAIAHRDLKSKNILVKKNGTCCIADLGLAVRHDSATDTIDIAPNHRVGTKRYMAPEVLDDSINMKHFESFKRADIYAMGLVFWEIARRCSIGGIHEDYQLPYYDLVPSDPSVEEMRKVVCEQKLRPNIPNRWQSCEALRVMAKIMRECWYANGAARLTALRIKKTLSQLSQQEG
3kcf	D	2.8	BS01	JZO	D	1	I211 K232 E245 Y249 L260 F262 S280 Y282 H283 L340	I41 K62 E75 Y79 L90 F92 S110 Y112 H113 L170	D333 K335 N338 D351 T375	D163 K165 N168 D181 T205	2.7.11.30	0004672,0004675,0005524,0006468,0007178,0016020				IC50=3690nM, Ki=35nM	P36897	19914068	4 	ISEGTTLKDLIYDMTTSGSGSGLPLLVQRTIARTIVLQESIGKGRFGEVWRGKWRGEEVAVKIFSSREERSWFREAEIYQTVMLRHENILGFIAADNKDNGTWTQLWLVSDYHEHGSLFDYLNRYTVTVEGMIKLALSTASGLAHLHMEIVGTQGKPAIAHRDLKSKNILVKKNGTCCIADLGLAVRHDSATDTIDIAPNHRVGTKRYMAPEVLDDSINMKHFESFKRADIYAMGLVFWEIARRCSIGGIHEDYQLPYYDLVPSDPSVEEMRKVVCEQKLRPNIPNRWQSCEALRVMAKIMRECWYANGAARLTALRIKKTLSQLSQQEG
3kcf	E	2.8	BS01	JZO	E	1	I211 A230 K232 Y249 L260 S280 Y282 H283 K337 L340	I41 A60 K62 Y79 L90 S110 Y112 H113 K167 L170	D333 K335 N338 D351 T375	D163 K165 N168 D181 T205	2.7.11.30	0004672,0004675,0005524,0006468,0007178,0016020				IC50=3690nM, Ki=35nM	P36897	19914068	5 	ISEGTTLKDLIYDMTTSGSGSGLPLLVQRTIARTIVLQESIGKGRFGEVWRGKWRGEEVAVKIFSSREERSWFREAEIYQTVMLRHENILGFIAADNKDNGTWTQLWLVSDYHEHGSLFDYLNRYTVTVEGMIKLALSTASGLAHLHMEIVGTQGKPAIAHRDLKSKNILVKKNGTCCIADLGLAVRHDSATDTIDIAPNHRVGTKRYMAPEVLDDSINMKHFESFKRADIYAMGLVFWEIARRCSIGGIHEDYQLPYYDLVPSDPSVEEMRKVVCEQKLRPNIPNRWQSCEALRVMAKIMRECWYANGAARLTALRIKKTLSQLSQQEG