6mod A 1.85 BS02 JWV A 1 M62 E77 T190 F191 M194 I197 G209 V216 H237 K238 D241 H264 M63 E78 T189 F190 M193 I196 G208 V215 H236 K237 D240 H263 3.5.1.108 0006796,0008759,0009245,0016787,0019637,0046872,0103117,1901135 ic50=0.71nM -logKd/Ki=9.15, IC50=0.71nM P47205 31283109 302 ATIKQRTLKNIIRATGVGLHSGEKVYLTLKPAPVDTGIVFCRTDLDPVVEIPARAENVGETTMSTTLVKGDVKVDTVEHLLSAMAGLGIDNAYVELSASEVPIMDGSAGPFVFLIQSAGLQEQEAAKKFVRIKREVSVEEGDKRAVFVPFDGFKVSFEIDFDHPVFRTQQASVDFSSTSFVKEVSRARTFGFMRDIEYLRSQNLALGGSVENAIVVDENRVLNEDGLRYEDEFVKHKILDAIGDLYLLGNSLIGEFRGFKSGHALNNQLLRTLIADKDAWEVVTFEDARTAPISYMRP