5qil A 1.98 BS01 J2V A 1 I211 K213 G214 V219 A230 K232 L260 S280 Y282 H283 G286 L340 D351 I15 K17 G18 V23 A34 K36 L64 S84 Y86 H87 G90 L144 D155 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 -logKd/Ki=11.52, IC50=0.003nM IC50=3.0nM P36897 30429955 601 GHMTIARDIVLQESIGKGRFGEVWRGKWRGEEVAVKIFSSREERSWFREAEIYQTVMLRHENILGFIAADNKDNGTWTQLWLVSDYHEHGSLFDYLNRYTVTVEGMIKLALSTASGLAHLHMEIVGTQGKPAIAHRDLKSKNILVKKNGTCCIADLGLAVRHDSATDTIDIAPNHRVGTKRYMAPEVLDDSINMKHFESFKRADIYAMGLVFWEIARRCSIGGIHEDYQLPYYDLVPSDPSVEEMRKVVCEQKLRPNIPNRWQSCEALRVMAKIMRECWYANGAARLTALRIKKTLSQLSQQE 5qin A 1.57 BS01 J2V A 1 V258 A275 K277 F294 L305 L323 T325 F327 H328 G331 L386 C396 D397 V19 A31 K33 F50 L61 L79 T81 F83 H84 G87 L142 C152 D153 D379 K381 N384 D397 T421 D135 K137 N140 D153 T175 2.7.11.30 0004672,0004675,0005524,0006468,0007178,0016020 -logKd/Ki=10.40, IC50=0.04nM IC50=40nM P37173 30429955 601 ELLPIELDTLVGKGRFAEVYKAKLKQFETVAVKIFPYEEYASWKTEKDIFSDINLKHENILQFLTAEERKTELGKQYWLITAFHAKGNLQEYLTRHVISWEDLRKLGSSLARGIAHLHSDHTPCGRPKMPIVHRDLKSSNILVKNDLTCCLCDFGLSLRLDPTLSVDDLANQVGTARYMAPEVLASAMNLENVESFKQTDVYSMALVLWEMTSRCNAVGEVKDYEPPFGSKVREHPCVASMADNVLADAGRPEIPSFWLNHQGIQMVCETLTECWDHDPEARLTAQCVAERFSEL