5jq8 A 1.94 BS01 I73 A 1 I10 G13 V18 A31 L83 H84 Q131 N132 L134 D145 I8 G11 V16 A29 L72 H73 Q120 N121 L123 D134 D127 K129 Q131 N132 D145 T165 D116 K118 Q120 N121 D134 T145 2.7.11.22 0000082,0000086,0000122,0000287,0000307,0000781,0000793,0000805,0000806,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005635,0005654,0005667,0005737,0005768,0005813,0005829,0005856,0006260,0006281,0006338,0006351,0006468,0006813,0007099,0007165,0007265,0007346,0008284,0010389,0010468,0015030,0016301,0016310,0018105,0019904,0030332,0031453,0031571,0032298,0035173,0043247,0043687,0045740,0045893,0046872,0051298,0051301,0051321,0071732,0090398,0097123,0097124,0097134,0097135,0097472,0106310,1905784 -logKd/Ki=5.70, Kd>2000nM IC50=580nM P24941 28125165 301 NFQKVEKIGEGTYGVVYKARNKLTGEVVALKKIPSTAIREISLLKELNHPNIVKLLDVIHTENKLYLVFEFLHQDLKKFMDASALTGIPLPLIKSYLFQLLQGLAFCHSHRVLHRDLKPQNLLINTEGAIKLADFGLARAFEVVTLWYRAPEILLGCKYYSTAVDIWSLGCIFAEMVTRRALFPGDSEIDQLFRIFRTLGTPDEVVWPGVTSMPDYKPSFPKWARQDFSKVVPPLDEDGRSLLSQMLHYDPNKRISAKAALAHPFFQDVTKPVPHLRL 8p77 J 1.8 BS01 I73 J 1 L18 A39 F91 M94 T96 D97 N141 N142 L144 L9 A24 F67 M70 T72 D73 N117 N118 L120 2.7.11.22,2.7.11.23 0000307,0000439,0001650,0001673,0004672,0004674,0004693,0005515,0005524,0005634,0005654,0005675,0005737,0005829,0005886,0006281,0006366,0006367,0006468,0008094,0008353,0016301,0016310,0042795,0045944,0048471,0050821,0051301,0051726,0070516,0070985,0106310,2000045 P50613 38480681 401 KRYEKLDFLGEGQFATVYKARIVAIKKKDGINRTALREIKLLQELSHPNIIGLLDAFGHKSNISLVFDFMETDLEVIIKDNSLVLTPSHIKAYMLMTLQGLEYLHQHWILHRDLKPNNLLLDENGVLKLADFGLAKSFGSPNRAYTHQVVTRWYRAPELLFGARMYGVGVDMWAVGCILAELLLRVPFLPGDSDLDQLTRIFETLGTPTEEQWPDMCSLPDYVTFKSFPGIPLHHIFSAAGDDLLDLIQGLFLFNPCARITATQALKMKYFSNRPGPTPGCQLPRP