3of8 A 2.2 BS01 I0Y A 1 Q20 C26 G62 E64 G69 L70 M71 A136 D163 H164 W190 Q20 C26 G62 E64 G69 L70 M71 A136 D163 H164 W190 Q20 C26 H164 N188 Q20 C26 H164 N188 3.4.22.15 0006508,0008234 -logKd/Ki=9.22, Ki=0.6nM P07711 20850545 501 EAPRSVDWREKGYVTPVKNQGQCGSCWAFSATGALEGQMFRKTGRLISLSEQNLVDCSGPQGNEGCNGGLMDYAFQYVQDNGGLDSEESYPYEATEESCKYNPKYSVANDTGFVDIPKQEKALMKAVATVGPISVAIDAGHESFLFYKEGIYFEPDCSSEDMDHGVLVVGYGFESTESDNNKYWLVKNSWGEEWGMGGYVKMAKDRRNHCGIASAASYPTV