2cvd A 1.45 BS02 HQL A 1 M11 G13 R14 M99 F102 W104 Y152 T159 M10 G12 R13 M98 F101 W103 Y151 T158 Y8 R14 R19 W104 Y7 R13 R18 W103 2.5.1.18,5.3.99.2 0000287,0001516,0004364,0004667,0005509,0005515,0005654,0005737,0005829,0006693,0007165,0007626,0009624,0010269,0016740,0016853,0042803,0043231,0046872,2000255 Kd=0.8uM -logKd/Ki=6.10, Kd=0.8uM IC50=3800nM O60760 16547010 2201 PNYKLTYFNMRGRAEIIRYIFAYLDIQYEDHRIEQADWPEIKSTLPFGKIPILEVDGLTLHQSLAIARYLTKNTDLAGNTEMEQCHVDAIVDTLDDFMSCFPWAEKKQDVKEQMFNELLTYNAPHLMQDLDTYLGGREWLIGMSVTWADFYWEICSTTLLVFKPDLLDNHPRLVTLRKKVQAIPAVANWIKRRPQTKL 2cvd B 1.45 BS02 HQL B 1 M11 G13 R14 M99 F102 W104 Y152 T159 L199 M10 G12 R13 M98 F101 W103 Y151 T158 L198 Y8 R14 R19 W104 Y7 R13 R18 W103 2.5.1.18,5.3.99.2 0000287,0001516,0004364,0004667,0005509,0005515,0005654,0005737,0005829,0006693,0007165,0007626,0009624,0010269,0016740,0016853,0042803,0043231,0046872,2000255 Kd=0.8uM IC50=3800nM O60760 16547010 2401 PNYKLTYFNMRGRAEIIRYIFAYLDIQYEDHRIEQADWPEIKSTLPFGKIPILEVDGLTLHQSLAIARYLTKNTDLAGNTEMEQCHVDAIVDTLDDFMSCFPWAEKKQDVKEQMFNELLTYNAPHLMQDLDTYLGGREWLIGMSVTWADFYWEICSTTLLVFKPDLLDNHPRLVTLRKKVQAIPAVANWIKRRPQTKL 2cvd C 1.45 BS02 HQL C 1 M11 G13 R14 M99 F102 W104 Y152 T159 M10 G12 R13 M98 F101 W103 Y151 T158 Y8 R14 R19 W104 Y7 R13 R18 W103 2.5.1.18,5.3.99.2 0000287,0001516,0004364,0004667,0005509,0005515,0005654,0005737,0005829,0006693,0007165,0007626,0009624,0010269,0016740,0016853,0042803,0043231,0046872,2000255 Kd=0.8uM IC50=3800nM O60760 16547010 2601 PNYKLTYFNMRGRAEIIRYIFAYLDIQYEDHRIEQADWPEIKSTLPFGKIPILEVDGLTLHQSLAIARYLTKNTDLAGNTEMEQCHVDAIVDTLDDFMSCFPWAEKKQDVKEQMFNELLTYNAPHLMQDLDTYLGGREWLIGMSVTWADFYWEICSTTLLVFKPDLLDNHPRLVTLRKKVQAIPAVANWIKRRPQTKL 2cvd D 1.45 BS02 HQL D 1 M11 G13 R14 M99 F102 W104 Y152 T159 M10 G12 R13 M98 F101 W103 Y151 T158 Y8 R14 R19 W104 Y7 R13 R18 W103 2.5.1.18,5.3.99.2 0000287,0001516,0004364,0004667,0005509,0005515,0005654,0005737,0005829,0006693,0007165,0007626,0009624,0010269,0016740,0016853,0042803,0043231,0046872,2000255 Kd=0.8uM IC50=3800nM O60760 16547010 2801 PNYKLTYFNMRGRAEIIRYIFAYLDIQYEDHRIEQADWPEIKSTLPFGKIPILEVDGLTLHQSLAIARYLTKNTDLAGNTEMEQCHVDAIVDTLDDFMSCFPWAEKKQDVKEQMFNELLTYNAPHLMQDLDTYLGGREWLIGMSVTWADFYWEICSTTLLVFKPDLLDNHPRLVTLRKKVQAIPAVANWIKRRPQTKL