2nq6 A 1.5 BS04 HM4 A 1 P192 Y195 Y196 C203 H212 H310 W353 P103 Y106 Y107 C114 H123 H221 W264 D229 D240 H303 H310 E336 E367 D140 D151 H214 H221 E247 E278 3.4.11.18 0006508,0070006 ic50=1.5uM -logKd/Ki=5.82, IC50=1.5uM EC50=>40000nM, IC50=400nM P53582 17114291 410 YRYTGKLRPHYPLMPTRPVPSYIQRPDYADHPLGMSESEQALKGTSQIKLLSSEDIEGMRLVCRLAREVLDVAAGMIKPGVTTEEIDHAVHLACIARNCYPSPLNYYNFPKSCCTSVNEVICHGIPDRRPLQEGDIVNVDITLYRNGYHGDLNETFFVGEVDDGARKLVQTTYECLMQAIDAVKPGVRYRELGNIIQKHAQANGFSVVRSYCGHGIHKLFHTAPNVPHYAKNKAVGVMKSGHVFTIEPMICEGGWQDETWPDGWTAVTRDGKRSAQFEHTLLVTDTGCEILTRRLDSARPHFMS