5twl A 2.42 BS01 H91 A 1 I17 K40 E57 C70 L86 E87 C89 E93 E136 L139 I149 D150 I18 K41 E58 C71 L87 E88 C90 E94 E137 L140 I150 D151 D132 K134 E136 N137 D150 S171 D133 K135 E137 N138 D151 S157 2.7.10.2,2.7.11.1 0004672,0004674,0005524,0006468 ic50=10.5nM -logKd/Ki=7.98, IC50=10.5nM Q14680 28926338 4000 GSKDYDELLKYYELHETIGTGGFAKVKLACHILTGEMVAIKIMDKNTLGSDLPRIKTEIEALKNLRHQHICQLYHVLETANKIFMVLEYCPGGELFDYIISQDRLSEEETRVVFRQIVSAVAYVHSQGYAHRDLKPENLLFDEYHKLKLIDFGLCGSLAYAAPELIQGKSYLGSEADVWSMGILLYVLMCGFLPFDDDNVMALYKKIMRGKYDVPKWLSPSSILLLQQMLQVDPKKRISMKNLLNHPWIMQDYNYPVEWQSKNPFIHLDDDCVTELSVHHRNNRQTMEDLISLWQYDHLTATYLLLLAKKARGKPVRLR