2fwz A 2.1 BS01 H71 A 1 N51 A55 M98 L107 F138 W162 N36 A40 M83 L92 F123 W147 3.6.4.10 0005524,0006457,0016887,0051082,0140662 ic50=50nM -logKd/Ki=7.30, IC50=50nM IC50=51nM, EC50=10.00nM P07900 16884307 1001 EVETFAFQAEIAQLMSLIINTFYSNKEIFLRELISNSSDALDKIRYESLTDPSKLDSGKELHINLIPNKQDRTLTIVDTGIGMTKADLINNLGTIAKSGTKAFMEALQAGADISMIGQFGVGFYSAYLVAEKVTVITKHNDDEQYAWESSAGGSFTVRTDTGEPMGRGTKVILHLKEDQTEYLEERRIKEIVKKHSQFIGYPITLFVE 4z1f A 2.703 BS01 H71 A 1 A123 I161 G162 M163 E167 N171 G202 F205 W231 T251 A55 I93 G94 M95 E99 N103 G104 F107 W133 T153 ? 0005524,0006457,0016887,0051082,0140662 IC50=205nM Q12931 25785725 1001 EPLHSIISSTESVQGSTSKHEFQAETKKLLDIVARSLYSEKEVFIRELISNASDALEKLRHKLVSDGQALPEMEIHLQTNAEKGTITIQDTGIGMTQEELVSNGVGFYSAFMVADRVEVYSRSAAPGSLGYQWLSDGSGVFEIAEASGVRTGTKIIIHLKSDCKEFSSEARVRDVVTKYSNFVSFPLYLNGRRMNTLQAIWMMDPKDVREWQHEEFYRYVAQAHDKPRYTLHYKTDAPLNIRSIFYVPDMKPSVALYSRKVLIQTKATDILPKWLRFIRGVVDSEDIPSALIRKLRDVLQQRLIKFFIDQSKKDAEKYAKFFEDYGLFMREGIVTATEQEVKEDIAKLLRYESSALPSGQLTSLSEYASRMRAGRNIYYLCAPNRHLAEHSPYYEAMKKKDTEVLFCFEQFDELTLLHLREFDKKKLISVET